Surendra Dawadi
Surendra Dawadi
Verified email at bcm.edu
Title
Cited by
Cited by
Year
Targeting Mycobacterium tuberculosis Biotin Protein Ligase (MtBPL) with Nucleoside-Based Bisubstrate Adenylation Inhibitors
MR Bockman, AS Kalinda, R Petrelli, T De la Mora-Rey, D Tiwari, F Liu, ...
Journal of medicinal chemistry 58 (18), 7349-7369, 2015
302015
Mutual potentiation drives synergy between trimethoprim and sulfamethoxazole
Y Minato, S Dawadi, SL Kordus, A Sivanandam, CC Aldrich, AD Baughn
Nature communications 9 (1), 1-7, 2018
282018
Synthesis and Pharmacokinetic Evaluation of Siderophore Biosynthesis Inhibitors for Mycobacterium tuberculosis
KM Nelson, K Viswanathan, S Dawadi, BP Duckworth, HI Boshoff, ...
Journal of medicinal chemistry 58 (14), 5459-5475, 2015
282015
Synthesis and pharmacological evaluation of nucleoside prodrugs designed to target siderophore biosynthesis in Mycobacterium tuberculosis
S Dawadi, S Kawamura, A Rubenstein, R Remmel, CC Aldrich
Bioorganic & medicinal chemistry 24 (6), 1314-1321, 2016
202016
Investigation and conformational analysis of fluorinated nucleoside antibiotics targeting siderophore biosynthesis
S Dawadi, K Viswanathan, HI Boshoff, CE Barry III, CC Aldrich
The Journal of organic chemistry 80 (10), 4835-4850, 2015
192015
Structure-based optimization of pyridoxal 5′-phosphate-dependent transaminase enzyme (BioA) inhibitors that target biotin biosynthesis in Mycobacterium tuberculosis
F Liu, S Dawadi, KM Maize, R Dai, SW Park, D Schnappinger, BC Finzel, ...
Journal of medicinal chemistry 60 (13), 5507-5520, 2017
182017
2-Aryl-8-aza-3-deazaadenosine analogues of 5′-O-[N-(salicyl) sulfamoyl] adenosine: nucleoside antibiotics that block siderophore biosynthesis in Mycobacterium tuberculosis
A Krajczyk, J Zeidler, P Januszczyk, S Dawadi, HI Boshoff, CE Barry III, ...
Bioorganic & medicinal chemistry 24 (14), 3133-3143, 2016
162016
Anchimerically activated ProTides as inhibitors of cap-dependent translation and inducers of chemosensitization in mantle cell lymphoma
A Okon, JJ Han, S Dawadi, C Demosthenous, CC Aldrich, M Gupta, ...
Journal of Medicinal Chemistry 60 (19), 8131-8144, 2017
152017
Targeting protein biotinylation enhances tuberculosis chemotherapy
D Tiwari, SW Park, MM Essawy, S Dawadi, A Mason, M Nandakumar, ...
Science translational medicine 10 (438), eaal1803, 2018
142018
Avoiding Antibiotic Inactivation in Mycobacterium tuberculosis by Rv3406 through Strategic Nucleoside Modification
MR Bockman, CA Engelhart, S Dawadi, P Larson, D Tiwari, DM Ferguson, ...
ACS infectious diseases 4 (7), 1102-1113, 2018
132018
Conformationally constrained cinnolinone nucleoside analogues as siderophore biosynthesis inhibitors for tuberculosis
S Dawadi, HIM Boshoff, SW Park, D Schnappinger, CC Aldrich
ACS medicinal chemistry letters 9 (4), 386-391, 2018
132018
Synthesis and analysis of bacterial folate metabolism intermediates and antifolates
S Dawadi, SL Kordus, AD Baughn, CC Aldrich
Organic letters 19 (19), 5220-5223, 2017
122017
Discovery of potent thrombin inhibitors from a protease-focused DNA-encoded chemical library
S Dawadi, N Simmons, G Miklossy, KM Bohren, JC Faver, MN Ucisik, ...
Proceedings of the National Academy of Sciences 117 (29), 16782-16789, 2020
42020
Chelating compounds and immobilized tethered chelators
RA Yokel, WR Harris, CD Spilling, RJ Kuhn, S Dawadi
US Patent 9,139,456, 2015
42015
Trapping hemiacetals with phosphono substituted palladium π-allyl complexes for the synthesis of substituted cyclic ethers
N Sutivisedsak, S Dawadi, CD Spilling
Tetrahedron letters 56 (23), 3534-3537, 2015
32015
Immobilized ligands for the removal of metal ions and methods thereof
C Spilling, W Harris, S Dawadi, B Hamper
32014
Optimization of guanidinylation of amines for the synthesis of protease-focused DNA-encoded chemical library
S Dawadi, N Simmons, M Matzuk
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 258, 2019
2019
Potentiation of para-aminosalicylic acid (PAS) by chemical inhibition of para-aminobenzoic acid (PABA) biosynthesis in Mycobacterium tuberculosis
S Dawadi, Y Minato, A Baughn, C Aldrich
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 255, 2018
2018
Synthesis and toxicological analysis of 5'sulfamoylated adenosine scaffolds for MtBPL drug development
M Fuller, M Bockman, S Dawadi, C Aldrich
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 253, 2017
2017
Avoiding antibiotic inactivation in Mycobacterium tuberculosis through strategic nucleoside modification
M Bockman, S Dawadi, C Aldrich
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 251, 2016
2016
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Articles 1–20