| 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological … P Minetti, MO Tinti, P Carminati, M Castorina, MA Di Cesare, S Di Serio, ... Journal of medicinal chemistry 48 (22), 6887-6896, 2005 | 110 | 2005 |
| Switchable reactivity of acylated α, β-dehydroamino ester in the Friedel− Crafts alkylation of indoles by changing the Lewis acid E Angelini, C Balsamini, F Bartoccini, S Lucarini, G Piersanti The Journal of Organic Chemistry 73 (14), 5654-5657, 2008 | 81 | 2008 |
| Synthesis of (E)-8-(3-Chlorostyryl)caffeine Analogues Leading to 9-Deazaxanthine Derivatives as Dual A2A Antagonists/MAO-B Inhibitors S Rivara, G Piersanti, F Bartoccini, G Diamantini, D Pala, T Riccioni, ... Journal of Medicinal Chemistry 56 (3), 1247-1261, 2013 | 60 | 2013 |
| Synthesis of (−)-Epi-Indolactam V by an intramolecular Buchwald–Hartwig C–N coupling cyclization reaction M Mari, F Bartoccini, G Piersanti The Journal of Organic Chemistry 78 (15), 7727-7734, 2013 | 58 | 2013 |
| A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole S Lucarini, F Bartoccini, F Battistoni, G Diamantini, G Piersanti, M Righi, ... Organic Letters 12 (17), 3844-3847, 2010 | 53 | 2010 |
| Iron-catalyzed direct C3-benzylation of indoles with benzyl alcohols through borrowing hydrogen G Di Gregorio, M Mari, F Bartoccini, G Piersanti The Journal of Organic Chemistry 82 (16), 8769-8775, 2017 | 47 | 2017 |
| Palladium (II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine … F Bartoccini, DM Cannas, F Fini, G Piersanti Organic letters 18 (11), 2762-2765, 2016 | 44 | 2016 |
| Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation S Bartolucci, F Bartoccini, M Righi, G Piersanti Organic letters 14 (2), 600-603, 2012 | 41 | 2012 |
| Synthesis of (±)-cis-Clavicipitic Acid by a Rh(I)-Catalyzed Intramolecular Imine Reaction F Bartoccini, M Casoli, M Mari, G Piersanti The Journal of Organic Chemistry 79 (7), 3255-3259, 2014 | 37 | 2014 |
| Synthesis of Boron‐and Silicon‐Containing Amino Acids through Copper‐Catalysed Conjugate Additions to Dehydroalanine Derivatives F Bartoccini, S Bartolucci, S Lucarini, G Piersanti European Journal of Organic Chemistry 2015 (15), 3352-3360, 2015 | 36 | 2015 |
| Organocatalytic synthesis of α-quaternary amino acid derivatives via aza-Friedel–Crafts alkylation of indoles with simple α-amidoacrylates M Righi, F Bartoccini, S Lucarini, G Piersanti Tetrahedron 67 (41), 7923-7928, 2011 | 36 | 2011 |
| A simple, modular synthesis of C4-substituted tryptophan derivatives F Bartoccini, S Bartolucci, M Mari, G Piersanti Organic & Biomolecular Chemistry 14, 10095-10110, 2016 | 34 | 2016 |
| Synthesis of benzo [1, 2-d; 3, 4-d′] diimidazole and 1H-pyrazolo [4, 3-b] pyridine as putative A 2A receptor antagonists G Piersanti, L Giorgi, F Bartoccini, G Tarzia, P Minetti, G Gallo, F Giorgi, ... Organic & Biomolecular Chemistry 5 (16), 2567-2571, 2007 | 28 | 2007 |
| C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology F Bartoccini, M Retini, G Piersanti Tetrahedron letters 61 (22), 151875, 2020 | 26 | 2020 |
| C4 Pictet–Spengler Reactions for the Synthesis of Core Structures in Hyrtiazepine Alkaloids T Abe, T Haruyama, K Yamada Synthesis 49 (18), 4141-4150, 2017 | 25 | 2017 |
| Development of a practical and sustainable strategy for the synthesis of ST1535 by an iron-catalyzed Kumada cross-coupling reaction F Bartoccini, G Piersanti, S Armaroli, A Cerri, W Cabri Tetrahedron Letters 55 (7), 1376-1378, 2014 | 23 | 2014 |
| Synthesis of 2-substituted tryptophans via a C3-to C2-alkyl migration M Mari, S Lucarini, F Bartoccini, G Piersanti, G Spadoni Beilstein Journal of Organic Chemistry 10 (1), 1991-1998, 2014 | 22 | 2014 |
| Synthesis and Biological Evaluation of Metabolites of 2-n-Butyl-9-methyl-8-[1, 2, 3] triazol-2-yl-9 H-purin-6-ylamine (ST1535), A Potent Antagonist of the A2A Adenosine … G Piersanti, F Bartoccini, S Lucarini, W Cabri, MA Stasi, T Riccioni, ... Journal of Medicinal Chemistry 56 (13), 5456-5463, 2013 | 22 | 2013 |
| Organocatalytic Aza-Friedel–Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho-and Benzofuranones Bearing a Quaternary Center at … F Bartoccini, M Mari, M Retini, S Bartolucci, G Piersanti The Journal of Organic Chemistry 83 (19), 12275-12283, 2018 | 19 | 2018 |
| Concise and convergent enantioselective total syntheses of (+)-and (−)-fumimycin M Retini, S Bartolucci, F Bartoccini, M Mari, G Piersanti The Journal of Organic Chemistry 84 (18), 12221-12227, 2019 | 18 | 2019 |
Giovanni PiersantiUniverità di Urbino Carlo Bo - Dipartimento di Scienze BiomolecolariEmail verificata su uniurb.it
