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Tommaso Felicetti
Tommaso Felicetti
Postdoc researcher, University of Perugia
Email verificata su unipg.it
Titolo
Citata da
Citata da
Anno
Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors
A Astolfi, T Felicetti, N Iraci, G Manfroni, S Massari, D Pietrella, O Tabarrini, ...
Journal of medicinal chemistry 60 (4), 1598-1604, 2017
662017
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction
T Felicetti, R Cannalire, D Pietrella, G Latacz, A Lubelska, G Manfroni, ...
Journal of medicinal chemistry 61 (17), 7827-7848, 2018
472018
Investigation on the effect of known potent S. aureus NorA efflux pump inhibitors on the staphylococcal biofilm formation
S Sabatini, M Piccioni, T Felicetti, S De Marco, G Manfroni, R Pagiotti, ...
RSC advances 7 (59), 37007-37014, 2017
362017
Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3‐Phenyl‐1,4‐benzothiazine Analogues
T Felicetti, R Cannalire, MS Burali, S Massari, G Manfroni, ML Barreca, ...
ChemMedChem 12 (16), 1293-1302, 2017
342017
Natural isoflavone biochanin A as a template for the design of new and potent 3-phenylquinolone efflux inhibitors against Mycobacterium avium
R Cannalire, D Machado, T Felicetti, SS Costa, S Massari, G Manfroni, ...
European Journal of Medicinal Chemistry 140, 321-330, 2017
312017
Modulating microRNA processing: enoxacin, the progenitor of a new class of drugs
T Felicetti, V Cecchetti, G Manfroni
Journal of Medicinal Chemistry 63 (21), 12275-12289, 2020
232020
Deciphering the Molecular Recognition Mechanism of Multidrug Resistance Staphylococcus aureus NorA Efflux Pump Using a Supervised Molecular Dynamics …
D Palazzotti, M Bissaro, G Bolcato, A Astolfi, T Felicetti, S Sabatini, ...
International journal of molecular sciences 20 (16), 4041, 2019
232019
Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions
R Cannalire, D Tarantino, G Piorkowski, T Carletti, S Massari, T Felicetti, ...
Antiviral Research 167, 6-12, 2019
232019
Broad‐spectrum flavivirus inhibitors: a medicinal chemistry point of view
T Felicetti, G Manfroni, V Cecchetti, R Cannalire
ChemMedChem 15 (24), 2391-2419, 2020
212020
From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors
S Massari, A Corona, S Distinto, J Desantis, A Caredda, S Sabatini, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 34 (1), 55-74, 2019
212019
Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation
A Astolfi, M Kudolo, J Brea, G Manni, G Manfroni, D Palazzotti, S Sabatini, ...
European Journal of Medicinal Chemistry 182, 111624, 2019
202019
Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position
T Felicetti, R Cannalire, MG Nizi, O Tabarrini, S Massari, ML Barreca, ...
European Journal of Medicinal Chemistry 155, 428-433, 2018
202018
Synthesis and characterization of 1, 2, 4-triazolo [1, 5-a] pyrimidine-2-carboxamide-based compounds targeting the PA-PB1 interface of influenza A virus polymerase
S Massari, C Bertagnin, MC Pismataro, A Donnadio, G Nannetti, ...
European journal of medicinal chemistry 209, 112944, 2021
192021
1, 2, 4-Triazolo [1, 5-a] pyrimidines: Efficient one-step synthesis and functionalization as influenza polymerase PA-PB1 interaction disruptors
MC Pismataro, T Felicetti, C Bertagnin, MG Nizi, A Bonomini, ML Barreca, ...
European Journal of Medicinal Chemistry 221, 113494, 2021
182021
Microbial efflux pump inhibitors: A journey around quinoline and indole derivatives
G Cernicchi, T Felicetti, S Sabatini
Molecules 26 (22), 6996, 2021
172021
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors
MG Nizi, J Desantis, Y Nakatani, S Massari, MA Mazzarella, G Shetye, ...
European Journal of Medicinal Chemistry 201, 112420, 2020
152020
C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors
T Felicetti, G Mangiaterra, R Cannalire, N Cedraro, D Pietrella, A Astolfi, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 35 (1), 584-597, 2020
142020
Discovery of 2-phenylquinolines with broad-spectrum anti-coronavirus activity
MG Nizi, L Persoons, A Corona, T Felicetti, G Cernicchi, S Massari, ...
ACS Medicinal Chemistry Letters 13 (5), 855-864, 2022
102022
Modifications on C6 and C7 positions of 3-phenylquinolone efflux pump inhibitors led to potent and safe antimycobacterial treatment adjuvants
T Felicetti, D Machado, R Cannalire, A Astolfi, S Massari, O Tabarrini, ...
ACS Infectious Diseases 5 (6), 982-1000, 2019
102019
Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors
R Cannalire, G Mangiaterra, T Felicetti, A Astolfi, N Cedraro, S Massari, ...
International Journal of Molecular Sciences 21 (19), 7037, 2020
82020
Il sistema al momento non può eseguire l'operazione. Riprova più tardi.
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