| Toll-like receptor 4 expression is increased in circulating mononuclear cells of patients with immunoglobulin A nephropathy R Coppo, R Camilla, A Amore, L Peruzzi, V Daprà, E Loiacono, S Vatrano, ... Clinical & Experimental Immunology 159 (1), 73-81, 2010 | 134 | 2010 |
| Homophymine A, an Anti-HIV Cyclodepsipeptide from the Sponge Homophymia sp. A Zampella, V Sepe, P Luciano, F Bellotta, MC Monti, MV D’Auria, ... The Journal of organic chemistry 73 (14), 5319-5327, 2008 | 127 | 2008 |
| Hijacking SARS-CoV-2/ACE2 receptor interaction by natural and semi-synthetic steroidal agents acting on functional pockets on the receptor binding domain A Carino, F Moraca, B Fiorillo, S Marchianò, V Sepe, M Biagioli, ... Frontiers in Chemistry 8, 572885, 2020 | 101 | 2020 |
| Design, synthesis, and biological evaluation of potent dual agonists of nuclear and membrane bile acid receptors C D’Amore, FS Di Leva, V Sepe, B Renga, C Del Gaudio, MV D’Auria, ... Journal of Medicinal Chemistry 57 (3), 937-954, 2014 | 97 | 2014 |
| Exploitation of cholane scaffold for the discovery of potent and selective farnesoid X receptor (FXR) and G-protein coupled bile acid receptor 1 (GP-BAR1) ligands C Festa, B Renga, C D’Amore, V Sepe, C Finamore, S De Marino, ... Journal of medicinal chemistry 57 (20), 8477-8495, 2014 | 85 | 2014 |
| Discovery that theonellasterol a marine sponge sterol is a highly selective FXR antagonist that protects against liver injury in cholestasis B Renga, A Mencarelli, C D'Amore, S Cipriani, MV D'Auria, V Sepe, ... PLoS One 7 (1), e30443, 2012 | 84 | 2012 |
| Farnesoid X receptor modulators 2014-present: a patent review V Sepe, E Distrutti, S Fiorucci, A Zampella Expert opinion on therapeutic patents 28 (5), 351-364, 2018 | 83 | 2018 |
| Solomonamides A and B, New Anti-inflammatory Peptides from Theonella swinhoei C Festa, S De Marino, V Sepe, MV D’Auria, G Bifulco, C Débitus, M Bucci, ... Organic Letters 13 (6), 1532-1535, 2011 | 81 | 2011 |
| Bile acid modulators for the treatment of nonalcoholic steatohepatitis (NASH) S Fiorucci, M Biagioli, V Sepe, A Zampella, E Distrutti Expert Opinion on Investigational Drugs 29 (6), 623-632, 2020 | 80 | 2020 |
| Discovery of sulfated sterols from marine invertebrates as a new class of marine natural antagonists of farnesoid-X-receptor V Sepe, G Bifulco, B Renga, C D’Amore, S Fiorucci, A Zampella Journal of medicinal chemistry 54 (5), 1314-1320, 2011 | 80 | 2011 |
| Modification on ursodeoxycholic acid (UDCA) scaffold. Discovery of bile acid derivatives as selective agonists of cell-surface G-protein coupled bile acid receptor 1 (GP-BAR1) V Sepe, B Renga, C Festa, C D’Amore, D Masullo, S Cipriani, FS Di Leva, ... Journal of medicinal chemistry 57 (18), 7687-7701, 2014 | 70 | 2014 |
| Perthamides C and D, two new potent anti-inflammatory cyclopeptides from a Solomon Lithistid sponge Theonella swinhoei C Festa, S De Marino, V Sepe, MC Monti, P Luciano, MV d'Auria, ... Tetrahedron 65 (50), 10424-10429, 2009 | 69 | 2009 |
| Isolation and structural elucidation of callipeltins J–M: antifungal peptides from the marine sponge Latrunculia sp. MV D'Auria, V Sepe, R D'Orsi, F Bellotta, C Debitus, A Zampella Tetrahedron 63 (1), 131-140, 2007 | 65 | 2007 |
| Homophymines B–E and A1–E1, a family of bioactive cyclodepsipeptides from the sponge Homophymia sp. A Zampella, V Sepe, F Bellotta, P Luciano, MV d'Auria, T Cresteil, ... Organic & biomolecular chemistry 7 (19), 4037-4044, 2009 | 62 | 2009 |
| Conicasterol E, a small heterodimer partner sparing farnesoid X receptor modulator endowed with a pregnane X receptor agonistic activity, from the marine sponge Theonella swinhoei V Sepe, R Ummarino, MV D’Auria, MG Chini, G Bifulco, B Renga, ... Journal of Medicinal Chemistry 55 (1), 84-93, 2012 | 59 | 2012 |
| Total synthesis and pharmacological characterization of solomonsterol A, a potent marine pregnane-X-receptor agonist endowed with anti-inflammatory activity V Sepe, R Ummarino, MV D’Auria, A Mencarelli, C D’Amore, B Renga, ... Journal of medicinal chemistry 54 (13), 4590-4599, 2011 | 59 | 2011 |
| Jaspamides M–P: new tryptophan modified jaspamide derivatives from the sponge Jaspis splendans F Gala, MV D'Auria, S De Marino, V Sepe, F Zollo, CD Smith, SN Keller, ... Tetrahedron 65 (1), 51-56, 2009 | 59 | 2009 |
| A nonuniform TFA homogenization technique based on piecewise interpolation functions of the inelastic field V Sepe, S Marfia, E Sacco International Journal of Solids and Structures 50 (5), 725-742, 2013 | 56 | 2013 |
| Concise synthesis of all stereoisomers of β-methoxytyrosine and determination of the absolute configuration of the residue in callipeltin A A Zampella, R D'Orsi, V Sepe, A Casapullo, MC Monti, MV D'Auria Organic Letters 7 (16), 3585-3588, 2005 | 55 | 2005 |
| Impaired itching perception in murine models of cholestasis is supported by dysregulation of GPBAR1 signaling S Cipriani, B Renga, C D’Amore, M Simonetti, AA De Tursi, A Carino, ... PLoS One 10 (7), e0129866, 2015 | 50 | 2015 |
Angela ZampellaProfessore di Chimica Organica, Federico IIEmail verificata su unina.it
