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Rosaria Gitto
Rosaria Gitto
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Pharmacophore‐based discovery of small‐molecule inhibitors of protein–protein interactions between HIV‐1 integrase and cellular cofactor LEDGF/p75
L De Luca, ML Barreca, S Ferro, F Christ, N Iraci, R Gitto, AM Monforte, ...
ChemMedChem 4 (8), 1311-1316, 2009
1372009
5H-[1, 2, 4] Oxadiazolo [5, 4-d][1, 5] benzothiazepines as anticonvulsant agents in DBA/2 mice
G De Sarro, A Chimirri, A De Sarro, R Gitto, S Grasso, M Zappalà
European journal of medicinal chemistry 30 (12), 925-929, 1995
1371995
1-Aryl-3,5-dihydro-4H-2,3-benzodiazepin-4-ones:  Novel AMPA Receptor Antagonists
A Chimirri, G De Sarro, A De Sarro, R Gitto, S Grasso, S Quartarone, ...
Journal of medicinal chemistry 40 (8), 1258-1269, 1997
1141997
Discovery of a novel and highly potent noncompetitive AMPA receptor antagonist
R Gitto, ML Barreca, L De Luca, G De Sarro, G Ferreri, S Quartarone, ...
Journal of medicinal chemistry 46 (1), 197-200, 2003
1012003
AMPA receptor antagonists as potential anticonvulsant drugs
GD Sarro, R Gitto, E Russo, GF Ibbadu, ML Barreca, LD Luca, A Chimirri
Current topics in medicinal chemistry 5 (1), 31-42, 2005
882005
GYKI 52466 and related 2, 3-benzodiazepines as anticonvulsant agents in DBA/2 mice
G De Sarro, A Chimirri, A De Sarro, R Gitto, S Grasso, P Giusti, ...
European journal of pharmacology 294 (2-3), 411-422, 1995
841995
Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor
L De Luca, S Ferro, R Gitto, ML Barreca, S Agnello, F Christ, Z Debyser, ...
Bioorganic & medicinal chemistry 18 (21), 7515-7521, 2010
812010
Synthesis and anticonvulsant properties of 2, 3, 3a, 4-tetrahydro-1H-pyrrolo [1, 2-a] benzimidazol-1-one derivatives
A Chimirri, A De Sarro, G De Sarro, R Gitto, M Zappala
Il Farmaco 56 (11), 821-826, 2001
792001
Comparative anticonvulsant activity of some 2, 3-benzodiazepine derivatives in rodents
G De Sarro, G Ferreri, P Gareri, E Russo, A De Sarro, R Gitto, A Chimirri
Pharmacology Biochemistry and Behavior 74 (3), 595-602, 2003
762003
Synthesis and evaluation of pharmacological properties of novel annelated 2, 3-benzodiazepine derivatives
R Gitto, V Orlando, S Quartarone, G De Sarro, A De Sarro, E Russo, ...
Journal of medicinal chemistry 46 (17), 3758-3761, 2003
712003
Synthesis and Evaluation of Pharmacological and Pharmacokinetic Properties of 11 H-[1, 2, 4] Triazolo [4, 5-c][2, 3] benzodiazepin-3 (2 H)-ones
M Zappala, R Gitto, F Bevacqua, S Quartarone, A Chimirri, M Rizzo, ...
Journal of medicinal chemistry 43 (25), 4834-4839, 2000
662000
New AMPA antagonists in epilepsy
E Russo, R Gitto, R Citraro, A Chimirri, G De Sarro
Expert opinion on investigational drugs 21 (9), 1371-1389, 2012
642012
3, 5-Dihydro-4 H-2, 3-benzodiazepine-4-thiones: a new class of AMPA receptor antagonists
A Chimirri, G De Sarro, A De Sarro, R Gitto, S Quartarone, M Zappalà, ...
Journal of medicinal chemistry 41 (18), 3409-3416, 1998
641998
Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as Potent Carbonic Anhydrase Inhibitors: Synthesis, Biological Evaluation, and Enzyme−Ligand X-ray …
R Gitto, S Agnello, S Ferro, L De Luca, D Vullo, J Brynda, P Mader, ...
Journal of medicinal chemistry 53 (6), 2401-2408, 2010
632010
HIV-1 integrase strand-transfer inhibitors: design, synthesis and molecular modeling investigation
L De Luca, S De Grazia, S Ferro, R Gitto, F Christ, Z Debyser, A Chimirri
European journal of medicinal chemistry 46 (2), 756-764, 2011
612011
Exploiting the 1-(4-fluorobenzyl) piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and …
L Ielo, B Deri, MP Germano, S Vittorio, S Mirabile, R Gitto, A Rapisarda, ...
European journal of medicinal chemistry 178, 380-389, 2019
592019
Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases
L De Luca, F Mancuso, S Ferro, MR Buemi, A Angeli, S Del Prete, ...
European journal of medicinal chemistry 143, 276-282, 2018
592018
Annelated 1, 5-benzodiazepines. I: Three, four, and five membered rings
A Chimirri, R Gitto, S Grasso, AM Monforte, G Romeo, M Zappala
Heterocycles (Sendai) 36 (3), 601-637, 1993
561993
Structure-based screening for the discovery of new carbonic anhydrase VII inhibitors
L De Luca, S Ferro, FM Damiano, CT Supuran, D Vullo, A Chimirri, R Gitto
European Journal of Medicinal Chemistry 71, 105-111, 2014
542014
Comparative anticonvulsant activity of N-acetyl-1-aryl-6, 7-dimethoxy-1, 2, 3, 4-tetrahydroisoquinoline derivatives in rodents
G Ferreri, A Chimirri, E Russo, R Gitto, P Gareri, A De Sarro, G De Sarro
Pharmacology Biochemistry and Behavior 77 (1), 85-94, 2004
542004
Il sistema al momento non può eseguire l'operazione. Riprova più tardi.
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