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Giovanni Piersanti
Giovanni Piersanti
Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari
Verified email at uniurb.it - Homepage
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Year
Cyclohexylcarbamic acid 3 ‘-or 4 ‘-substituted biphenyl-3-yl esters as fatty acid amide hydrolase inhibitors: synthesis, quantitative structure− activity relationships, and …
M Mor, S Rivara, A Lodola, PV Plazzi, G Tarzia, A Duranti, A Tontini, ...
Journal of medicinal chemistry 47 (21), 4998-5008, 2004
3282004
Design, synthesis, and structure− activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors
G Tarzia, A Duranti, A Tontini, G Piersanti, M Mor, S Rivara, PV Plazzi, ...
Journal of medicinal chemistry 46 (12), 2352-2360, 2003
2092003
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological …
P Minetti, MO Tinti, P Carminati, M Castorina, MA Di Cesare, S Di Serio, ...
Journal of medicinal chemistry 48 (22), 6887-6896, 2005
1092005
Enantioselective Total Synthesis of (−)‐Acylfulvene and (−)‐Irofulven
M Movassaghi, G Piizzi, DS Siegel, G Piersanti
Angewandte Chemie 118 (35), 5991-5995, 2006
842006
Switchable reactivity of acylated α, β-dehydroamino ester in the Friedel− Crafts alkylation of indoles by changing the Lewis acid
E Angelini, C Balsamini, F Bartoccini, S Lucarini, G Piersanti
The Journal of Organic Chemistry 73 (14), 5654-5657, 2008
812008
Synthesis and quantitative structure− activity relationship of fatty acid amide hydrolase inhibitors: Modulation at the N-portion of biphenyl-3-yl alkylcarbamates
M Mor, A Lodola, S Rivara, F Vacondio, A Duranti, A Tontini, S Sanchini, ...
Journal of medicinal chemistry 51 (12), 3487-3498, 2008
762008
Synthesis of tryptamine derivatives via a direct, one-pot reductive alkylation of indoles
M Righi, F Topi, S Bartolucci, A Bedini, G Piersanti, G Spadoni
The Journal of Organic Chemistry 77 (14), 6351-6357, 2012
742012
Synthesis and structure–activity relationships of FAAH inhibitors: cyclohexylcarbamic acid biphenyl esters with chemical modulation at the proximal phenyl ring
G Tarzia, A Duranti, G Gatti, G Piersanti, A Tontini, S Rivara, A Lodola, ...
ChemMedChem: Chemistry Enabling Drug Discovery 1 (1), 130-139, 2006
732006
Iridium-catalyzed direct synthesis of tryptamine derivatives from indoles: exploiting N-protected β-amino alcohols as alkylating agents
S Bartolucci, M Mari, A Bedini, G Piersanti, G Spadoni
The Journal of Organic Chemistry 80 (6), 3217-3222, 2015
642015
Enantioselective total synthesis of (−)-Acylfulvene and (−)-Irofulven
DS Siegel, G Piizzi, G Piersanti, M Movassaghi
The Journal of organic chemistry 74 (24), 9292-9304, 2009
632009
Synthesis of (E)-8-(3-Chlorostyryl)caffeine Analogues Leading to 9-Deazaxanthine Derivatives as Dual A2A Antagonists/MAO-B Inhibitors
S Rivara, G Piersanti, F Bartoccini, G Diamantini, D Pala, T Riccioni, ...
Journal of Medicinal Chemistry 56 (3), 1247-1261, 2013
602013
Quantifying amino acid conformational preferences and side-chain–side-chain interactions in β-hairpins
ST Phillips, G Piersanti, PA Bartlett
Proceedings of the National Academy of Sciences 102 (39), 13737-13742, 2005
592005
Synthesis of (−)-Epi-Indolactam V by an intramolecular Buchwald–Hartwig C–N coupling cyclization reaction
M Mari, F Bartoccini, G Piersanti
The Journal of Organic Chemistry 78 (15), 7727-7734, 2013
552013
A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole
S Lucarini, F Bartoccini, F Battistoni, G Diamantini, G Piersanti, M Righi, ...
Organic Letters 12 (17), 3844-3847, 2010
512010
Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen
G Di Gregorio, M Mari, F Bartoccini, G Piersanti
The Journal of Organic Chemistry 82 (16), 8769-8775, 2017
472017
A Trans-Stereoselective Synthesis of 3-Halo-4-alkyl (aryl)-NH-azetidin-2-ones
E Bandini, G Favi, G Martelli, M Panunzio, G Piersanti
Organic Letters 2 (8), 1077-1079, 2000
472000
Tricyclic alkylamides as melatonin receptor ligands with antagonist or inverse agonist activity
V Lucini, M Pannacci, F Scaglione, F Fraschini, S Rivara, M Mor, F Bordi, ...
Journal of medicinal chemistry 47 (17), 4202-4212, 2004
432004
Palladium (II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine …
F Bartoccini, DM Cannas, F Fini, G Piersanti
Organic letters 18 (11), 2762-2765, 2016
422016
Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation
S Bartolucci, F Bartoccini, M Righi, G Piersanti
Organic letters 14 (2), 600-603, 2012
402012
New branched macrocyclic ligand and its side-arm, two urea-based receptors for anions: synthesis, binding studies and crystal structure
M Formica, V Fusi, E Macedi, P Paoli, G Piersanti, P Rossi, G Zappia, ...
New Journal of Chemistry 32 (7), 1204-1214, 2008
402008
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