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Dritan Hasa
Dritan Hasa
Department of Chemical and Pharmaceutical Sciences, University of Trieste
Email verificata su units.it - Home page
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Citata da
Anno
Cocrystal formation through mechanochemistry: from neat and liquid‐assisted grinding to polymer‐assisted grinding
D Hasa, G Schneider Rauber, D Voinovich, W Jones
Angewandte Chemie 127 (25), 7479-7483, 2015
2692015
Screening for new pharmaceutical solid forms using mechanochemistry: A practical guide
D Hasa, W Jones
Advanced drug delivery reviews 117, 147-161, 2017
1892017
Mechanochemical synthesis of multicomponent crystals: One liquid for one polymorph? A myth to dispel
D Hasa, E Miniussi, W Jones
Crystal Growth & Design 16 (8), 4582-4588, 2016
1302016
Polymer-assisted grinding, a versatile method for polymorph control of cocrystallization
D Hasa, E Carlino, W Jones
Crystal Growth & Design 16 (3), 1772-1779, 2016
1022016
Oral bioavailability of silymarin phytocomplex formulated as self-emulsifying pellets
T Iosio, D Voinovich, B Perissutti, F Serdoz, D Hasa, I Grabnar, ...
Phytomedicine 18 (6), 505-512, 2011
692011
Selective synthesis of a salt and a cocrystal of the ethionamide–salicylic acid system
D Bernasconi, S Bordignon, F Rossi, E Priola, C Nervi, R Gobetto, ...
Crystal Growth & Design 20 (2), 906-915, 2019
562019
A new soluble and bioactive polymorph of praziquantel
D Zanolla, B Perissutti, N Passerini, MR Chierotti, D Hasa, D Voinovich, ...
European Journal of Pharmaceutics and Biopharmaceutics 127, 19-28, 2018
542018
A new approach to enhance oral bioavailability of Silybum Marianum dry extract: Association of mechanochemical activation and spray congealing
N Passerini, B Perissutti, B Albertini, E Franceschinis, D Lenaz, D Hasa, ...
Phytomedicine 19 (2), 160-168, 2012
482012
Drug salt formation via mechanochemistry: the case study of vincamine
D Hasa, B Perissutti, C Cepek, S Bhardwaj, E Carlino, M Grassi, ...
Molecular Pharmaceutics 10 (1), 211-224, 2013
432013
Enhanced Oral Bioavailability of Vinpocetine Through Mechanochemical Salt Formation: Physico-Chemical Characterization and In Vivo Studies
D Hasa, D Voinovich, B Perissutti, M Grassi, A Bonifacio, V Sergo, ...
Pharmaceutical research 28, 1870-1883, 2011
372011
Reduction of melting temperature and enthalpy of drug crystals: theoretical aspects
D Hasa, D Voinovich, B Perissutti, G Grassi, S Fiorentino, R Farra, ...
European Journal of Pharmaceutical Sciences 50 (1), 17-28, 2013
362013
Rationale of using Vinca minor Linne dry extract phytocomplex as a vincamine’s oral bioavailability enhancer
D Hasa, B Perissutti, S Dall’Acqua, MR Chierotti, R Gobetto, I Grabnar, ...
European Journal of Pharmaceutics and Biopharmaceutics 84 (1), 138-144, 2013
332013
Mechanochemical reactivity inhibited, prohibited and reversed by liquid additives: examples from crystal-form screens
M Arhangelskis, DK Bučar, S Bordignon, MR Chierotti, SA Stratford, ...
Chemical Science 12 (9), 3264-3269, 2021
292021
Multidisciplinary approach on characterizing a mechanochemically activated composite of vinpocetine and crospovidone
D Hasa, D Voinovich, B Perissutti, A Bonifacio, M Grassi, E Franceschinis, ...
Journal of pharmaceutical sciences 100 (3), 915-932, 2011
282011
Mechanochemical formation of racemic praziquantel hemihydrate with improved biopharmaceutical properties
D Zanolla, D Hasa, M Arhangelskis, G Schneider-Rauber, MR Chierotti, ...
Pharmaceutics 12 (3), 289, 2020
272020
Development and pharmacokinetic evaluation of erythromycin lipidic formulations for oral administration in rainbow trout (Oncorhynchus mykiss)
F Serdoz, D Voinovich, B Perissutti, I Grabnar, D Hasa, R Ballestrazzi, ...
European journal of pharmaceutics and biopharmaceutics 78 (3), 401-407, 2011
232011
Exploring the shape influence on melting temperature, enthalpy, and solubility of organic drug nanocrystals by a thermodynamic model
G Chiarappa, A Piccolo, I Colombo, D Hasa, D Voinovich, M Moneghini, ...
Crystal Growth & Design 17 (8), 4072-4083, 2017
212017
Simultaneous release and ADME processes of poorly water-soluble drugs: mathematical modeling
G Grassi, D Hasa, D Voinovich, B Perissutti, B Dapas, R Farra, ...
Molecular Pharmaceutics 7 (5), 1488-1497, 2010
212010
Drug nanocrystals: theoretical background of solubility increase and dissolution rate enhancement
D Hasa, B Perissutti, D Voinovich, M Abrami, R Farra, SM Fiorentino, ...
Chemical and Biochemical Engineering Quarterly 28 (3), 247-258, 2014
202014
A physiologically-oriented mathematical model for the description of in vivo drug release and absorption
R Del Cont, M Abrami, D Hasa, B Perissutti, D Voinovich, A Barba, ...
ADMET and DMPK 2 (2), 80-97, 2014
192014
Il sistema al momento non può eseguire l'operazione. Riprova più tardi.
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