Marco Radi
Title
Cited by
Cited by
Year
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: part 2. Synthesis of rigid pyrazolones
D Castagnolo, F Manetti, M Radi, B Bechi, M Pagano, A De Logu, ...
Bioorganic & medicinal chemistry 17 (15), 5716-5721, 2009
1672009
Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis
D Castagnolo, A De Logu, M Radi, B Bechi, F Manetti, M Magnani, ...
Bioorganic & medicinal chemistry 16 (18), 8587-8591, 2008
1352008
ATP-competitive inhibitors of mTOR: an update
S Schenone, C Brullo, F Musumeci, M Radi, M Botta
Current medicinal chemistry 18 (20), 2995-3014, 2011
1272011
Vascular endothelial growth factor (VEGF) receptors: drugs and new inhibitors
F Musumeci, M Radi, C Brullo, S Schenone
Journal of medicinal chemistry 55 (24), 10797-10822, 2012
1262012
Biologically Driven Synthesis of Pyrazolo[3,4-d]pyrimidines As Protein Kinase Inhibitors: An Old Scaffold As a New Tool for Medicinal Chemistry and Chemical …
S Schenone, M Radi, F Musumeci, C Brullo, M Botta
Chemical reviews 114 (14), 7189-7238, 2014
862014
Microwave-assisted organocatalytic multicomponent Knoevenagel/hetero Diels–Alder reaction for the synthesis of 2, 3-dihydropyran [2, 3-c] pyrazoles
M Radi, V Bernardo, B Bechi, D Castagnolo, M Pagano, M Botta
Tetrahedron Letters 50 (47), 6572-6575, 2009
862009
Toward the discovery of novel anti‐HIV drugs. Second‐generation inhibitors of the cellular ATPase DDX3 with improved anti‐HIV activity: Synthesis, structure–activity …
G Maga, F Falchi, M Radi, L Botta, G Casaluce, M Bernardini, H Irannejad, ...
ChemMedChem 6 (8), 1371-1389, 2011
802011
Discovery of the first small molecule inhibitor of human DDX3 specifically designed to target the RNA binding site: towards the next generation HIV-1 inhibitors
M Radi, F Falchi, A Garbelli, A Samuele, V Bernardo, S Paolucci, ...
Bioorganic & medicinal chemistry letters 22 (5), 2094-2098, 2012
782012
Microwave-enhanced Sonogashira coupling reaction of substituted pyrimidinones and pyrimidine nucleosides
E Petricci, M Radi, F Corelli, M Botta
Tetrahedron letters 44 (51), 9181-9184, 2003
782003
Design, Synthesis, Biological Activity, and ADME Properties of Pyrazolo[3,4-d]pyrimidines Active in Hypoxic Human Leukemia Cells: A Lead Optimization Study
M Radi, E Dreassi, C Brullo, E Crespan, C Tintori, V Bernardo, M Valoti, ...
Journal of medicinal chemistry 54 (8), 2610-2626, 2011
702011
Recent highlights in the synthesis of highly functionalized pyrimidines
M Radi, S Schenone, M Botta
Organic & biomolecular chemistry 7 (14), 2841-2847, 2009
692009
Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis
D Castagnolo, M Radi, F Dessì, F Manetti, M Saddi, R Meleddu, ...
Bioorganic & medicinal chemistry letters 19 (8), 2203-2205, 2009
642009
Discovery and SAR of 1, 3, 4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents
M Radi, E Crespan, G Botta, F Falchi, G Maga, F Manetti, V Corradi, ...
Bioorganic & medicinal chemistry letters 18 (3), 1207-1211, 2008
632008
Targeting the human DEAD-box polypeptide 3 (DDX3) RNA helicase as a novel strategy to inhibit viral replication
A Garbelli, M Radi, F Falchi, S Beermann, S Zanoli, F Manetti, U Dietrich, ...
Current medicinal chemistry 18 (20), 3015-3027, 2011
562011
New insights into small‐molecule inhibitors of Bcr‐Abl
S Schenone, O Bruno, M Radi, M Botta
Medicinal research reviews 31 (1), 1-41, 2011
542011
Microwave-assisted acylation of amines, alcohols, and phenols by the use of solid-supported reagents (SSRs)
E Petricci, C Mugnaini, M Radi, F Corelli, M Botta
The Journal of organic chemistry 69 (23), 7880-7887, 2004
502004
Discovery of Chiral Cyclopropyl Dihydro-Alkylthio-Benzyl-Oxopyrimidine (S-DABO) Derivatives as Potent HIV-1 Reverse Transcriptase Inhibitors with High Activity …
M Radi, G Maga, M Alongi, L Angeli, A Samuele, S Zanoli, L Bellucci, ...
Journal of medicinal chemistry 52 (3), 840-851, 2009
492009
Practical one-pot two-step protocol for the microwave-assisted synthesis of highly functionalized rhodanine derivatives
M Radi, L Botta, G Casaluce, M Bernardini, M Botta
Journal of combinatorial chemistry 12 (1), 200-205, 2010
482010
HIV-1 RT inhibitors with a novel mechanism of action: NNRTIs that compete with the nucleotide substrate
G Maga, M Radi, MA Gerard, M Botta, E Ennifar
Viruses 2 (4), 880-899, 2010
462010
Discovery of multitarget antivirals acting on both the Dengue virus NS5-NS3 interaction and the host Src/Fyn kinases
P Vincetti, F Caporuscio, S Kaptein, A Gioiello, V Mancino, Y Suzuki, ...
Journal of medicinal chemistry 58 (12), 4964-4975, 2015
432015
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