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Jon Merlin
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Quantification of functional selectivity at the human α1A-adrenoceptor
BA Evans, N Broxton, J Merlin, M Sato, DS Hutchinson, A Christopoulos, ...
Molecular pharmacology 79 (2), 298-307, 2011
912011
Adrenoceptors in white, brown, and brite adipocytes
BA Evans, J Merlin, T Bengtsson, DS Hutchinson
British journal of pharmacology 176 (14), 2416-2432, 2019
592019
Could burning fat start with a brite spark? Pharmacological and nutritional ways to promote thermogenesis
J Merlin, BA Evans, N Dehvari, M Sato, T Bengtsson, DS Hutchinson
Molecular nutrition & food research 60 (1), 18-42, 2016
552016
The PPARγ agonist rosiglitazone promotes the induction of brite adipocytes, increasing β-adrenoceptor-mediated mitochondrial function and glucose uptake
J Merlin, M Sato, C Nowell, M Pakzad, R Fahey, J Gao, N Dehvari, ...
Cellular signalling 42, 54-66, 2018
482018
The M3-muscarinic acetylcholine receptor stimulates glucose uptake in L6 skeletal muscle cells by a CaMKK–AMPK–dependent mechanism
J Merlin, BA Evans, RI Csikasz, T Bengtsson, RJ Summers, ...
Cellular signalling 22 (7), 1104-1113, 2010
472010
β2‐Adrenoceptors increase translocation of GLUT4 via GPCR kinase sites in the receptor C‐terminal tail
N Dehvari, DS Hutchinson, J Nevzorova, OS Dallner, M Sato, M Kocan, ...
British journal of pharmacology 165 (5), 1442-1456, 2012
362012
Factors influencing biased agonism in recombinant cells expressing the human α1A‐adrenoceptor
ED da Silva Junior, M Sato, J Merlin, N Broxton, DS Hutchinson, ...
British journal of pharmacology 174 (14), 2318-2333, 2017
342017
α2‐Adrenoceptors activate noradrenaline‐mediated glycogen turnover in chick astrocytes
DS Hutchinson, SL Catus, J Merlin, RJ Summers, ME Gibbs
Journal of neurochemistry 117 (5), 915-926, 2011
312011
Rosiglitazone and a β3-adrenoceptor agonist are both required for functional browning of white adipocytes in culture
J Merlin, M Sato, RJ Summers, BA Evans, DS Hutchinson
Frontiers in endocrinology 9, 357384, 2018
272018
BRL37344 stimulates GLUT4 translocation and glucose uptake in skeletal muscle via β2-adrenoceptors without causing classical receptor desensitization
S Mukaida, M Sato, AI Öberg, N Dehvari, JM Olsen, M Kocan, ML Halls, ...
American Journal of Physiology-Regulatory, Integrative and Comparative …, 2019
192019
Orthosteric Binding of ρ-Da1a, a Natural Peptide of Snake Venom Interacting Selectively with the α1A-Adrenoceptor
A Maďga, J Merlin, E Marcon, C Rouget, M Larregola, B Gilquin, ...
PLoS One 8 (7), e68841, 2013
132013
The metabolic effects of mirabegron are mediated primarily by β3‐adrenoceptors
N Dehvari, M Sato, MH Bokhari, A Kalinovich, S Ham, J Gao, ...
Pharmacology Research & Perspectives 8 (5), e00643, 2020
102020
Multipathway In vitro pharmacological characterization of specialized proresolving G protein-coupled receptors
J Merlin, J Park, TH Vandekolk, SA Fabb, J Allinne, RJ Summers, ...
Molecular Pharmacology 101 (4), 246-256, 2022
92022
Pharmacological insights into safety and efficacy determinants for the development of adenosine receptor biased agonists in the treatment of heart failure
P Rueda, J Merlin, S Chimenti, PJ White, A Christopoulos, RJ Summers, ...
Frontiers in Pharmacology 12, 628060, 2021
92021
Implications of ligand-receptor binding kinetics on GLP-1R signalling
P Zhao, TT Truong, J Merlin, PM Sexton, D Wootten
Biochemical Pharmacology 199, 114985, 2022
72022
Deletion of GPR21 improves glucose homeostasis and inhibits the CCL2-CCR2 axis by divergent mechanisms
DM Riddy, HL Kammoun, AJ Murphy, S Bosnyak-Gladovic, ...
BMJ Open Diabetes Research and Care 9 (2), e002285, 2021
52021
Effects of hypoxia-ischemia and inotropes on expression of cardiac adrenoceptors in the preterm fetal sheep
DS Hutchinson, N Brew, T Vu, J Merlin, N Hale, DW Walker, FY Wong
Journal of Applied Physiology 125 (5), 1368-1377, 2018
42018
Similar drugs can produce surprisingly different results
ED da Silva Junior, M Sato, J Merlin, N Broxton, DS Hutchinson, S Ventur, ...
2019
Metabolic effects of mirabegron in primary adipocytes in vitro, and on metabolic parameters in vivo
D Hutchinson, N Dehvari, M Sato, W Gao, L Whiting, A Kalinovich, ...
2019
Metabolic effects of mirabegron in mice: implications for use in diabetes
DS Hutchinson, N Dehvari, M Sato, J Gao, L Whiting, S Mukaida, J Merlin, ...
Proceedings for Annual Meeting of The Japanese Pharmacological Society …, 2018
2018
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Articles 1–20