| Synthesis and biological evaluation (in vitro and in vivo) of cyclic arginine–glycine–aspartate (RGD) peptidomimetic–paclitaxel conjugates targeting integrin αVβ3 R Colombo, M Mingozzi, L Belvisi, D Arosio, U Piarulli, N Carenini, ... American Chemical Society, 2012 | 91 | 2012 |
| Cyclic RGD peptidomimetics containing bifunctional diketopiperazine scaffolds as new potent integrin ligands M Marchini, M Mingozzi, R Colombo, I Guzzetti, L Belvisi, F Vasile, ... Chemistry–A European Journal 18 (20), 6195-6207, 2012 | 89 | 2012 |
| PhthalaPhos: Chiral supramolecular ligands for enantioselective rhodium-catalyzed hydrogenation reactions L Pignataro, S Carboni, M Civera, R Colombo, U Piarulli, C Gennari Angew. Chem. Int. Ed 49 (37), 6633-6637, 2010 | 69 | 2010 |
| Structure–activity study of bioisosteric trifluoromethyl and pentafluorosulfanyl indole inhibitors of the AAA ATPase p97 C Alverez, MR Arkin, SL Bulfer, R Colombo, M Kovaliov, MG LaPorte, ... ACS medicinal chemistry letters 6 (12), 1225-1230, 2015 | 57 | 2015 |
| The therapeutic window of antibody drug conjugates: a dogma in need of revision R Colombo, JR Rich Cancer Cell 40 (11), 1255-1263, 2022 | 54 | 2022 |
| General and Chemoselective N‐Transacylation of Secondary Amides by Means of Perfluorinated Anhydrides P Rota, P Allevi, R Colombo, ML Costa, M Anastasia Angewandte Chemie 122 (10), 1894-1897, 2010 | 44 | 2010 |
| Total synthesis and biological evaluation of tubulysin analogues R Colombo, Z Wang, J Han, R Balachandran, HN Daghestani, ... The Journal of Organic Chemistry 81 (21), 10302-10320, 2016 | 37 | 2016 |
| Optimization of pyrazole-containing 1, 2, 4-triazolo-[3, 4-b] thiadiazines, a new class of STAT3 pathway inhibitors MG LaPorte, Z Wang, R Colombo, A Garzan, VA Peshkov, M Liang, ... Bioorganic & medicinal chemistry letters 26 (15), 3581-3585, 2016 | 31 | 2016 |
| Microwave-assisted cyclization of unprotected dipeptides in water to 2, 5-piperazinediones and self-assembly study of products and reagents M Kurbasic, S Semeraro, AM Garcia, S Kralj, E Parisi, C Deganutti, ... Synthesis 51 (14), 2829-2838, 2019 | 29 | 2019 |
| Chemoselective synthesis of sialic acid 1, 7-lactones P Allevi, P Rota, R Scaringi, R Colombo, M Anastasia The Journal of organic chemistry 75 (16), 5542-5548, 2010 | 28 | 2010 |
| The first synthesis of N-acetylneuraminic acid 1, 7-lactone R Colombo, M Anastasia, P Rota, P Allevi Chemical communications, 5517-5519, 2008 | 21 | 2008 |
| PTPRT epigenetic silencing defines lung cancer with STAT3 activation and can direct STAT3 targeted therapies M Sen, A Kindsfather, L Danilova, F Zhang, R Colombo, MG LaPorte, ... Epigenetics 15 (6-7), 604-617, 2020 | 20 | 2020 |
| Optimization of phenyl indole inhibitors of the AAA+ ATPase p97 MG LaPorte, JC Burnett, R Colombo, SL Bulfer, C Alverez, TF Chou, ... ACS medicinal chemistry letters 9 (11), 1075-1081, 2018 | 20 | 2018 |
| Combination of a binaphthol-derived phosphite and a C 1-symmetric phosphinamine generates heteroleptic catalysts in Rh-and Pd-mediated reactions L Pignataro, B Lynikaite, R Colombo, S Carboni, M Krupička, U Piarulli, ... Chemical communications, 3539-3541, 2009 | 18 | 2009 |
| Asymmetric total synthesis and biological evaluation of (+)-cycloclavine SR McCabe, P Wipf Synthesis 51 (01), 213-224, 2019 | 16 | 2019 |
| Metabolite-Based Modification of Poly(l-lysine) for Improved Gene Delivery MA Urello, L Xiang, R Colombo, A Ma, A Joseph, J Boyd, N Peterson, ... Biomacromolecules 21 (9), 3596-3607, 2020 | 14 | 2020 |
| A threonine turnstile defines a dynamic amphiphilic binding motif in the AAA ATPase p97 allosteric binding site JC Burnett, C Lim, BD Peyser, LP Samankumara, M Kovaliov, R Colombo, ... Organic & biomolecular chemistry 15 (19), 4096-4114, 2017 | 14 | 2017 |
| Selective O-acylation of unprotected N-benzylserine methyl ester and O, N-acyl transfer in the formation of cyclo [Asp-Ser] diketopiperazines M Marchini, M Mingozzi, R Colombo, C Gennari, M Durini, U Piarulli Tetrahedron 66 (49), 9528-9531, 2010 | 11 | 2010 |
| Elucidation of the opening of the epoxidic ring of the 3β-acetoxy-14α, 15α-epoxy-5α-cholest-8-en-7-one by methanol, using NMR techniques assisted by a conformational study … M Anastasia, P Allevi, R Colombo, E Giannini Steroids 72 (11-12), 809-818, 2007 | 8 | 2007 |
| Engineered Ultrasmall Nanoparticle Drug‐Immune Conjugates with “Hit and Run” Tumor Delivery to Eradicate Gastric Cancer L Zhang, V Aragon‐Sanabria, A Aditya, M Marelli, T Cao, F Chen, B Yoo, ... Advanced therapeutics 6 (3), 2200209, 2023 | 7 | 2023 |
