| Total synthesis and structural confirmation of the marine natural product Dysinosin A: a novel inhibitor of thrombin and Factor VIIa S Hanessian, R Margarita, A Hall, S Johnstone, M Tremblay, L Parlanti Journal of the American Chemical Society 124 (45), 13342-13343, 2002 | 121 | 2002 |
| A general method for the α-acyloxylation of carbonyl compounds CS Beshara, A Hall, RL Jenkins, KL Jones, TC Jones, NM Killeen, ... Organic letters 7 (25), 5729-5732, 2005 | 109 | 2005 |
| Non-acidic pyrazole EP1 receptor antagonists with in vivo analgesic efficacy A Hall, A Billinton, SH Brown, NM Clayton, A Chowdhury, GMP Giblin, ... Bioorganic & medicinal chemistry letters 18 (11), 3392-3399, 2008 | 96 | 2008 |
| One-Pot, Three-Component Sulfonimidamide Synthesis Exploiting the Sulfinylamine Reagent N-Sulfinyltritylamine, TrNSO MCW Thomas Q. Davies, Adrian Hall Angewandte Chemie 129, 15133-15137, 2017 | 78* | 2017 |
| Copper-catalyzed coupling of hydroxylamines with aryl iodides KL Jones, A Porzelle, A Hall, MD Woodrow, NCO Tomkinson Organic letters 10 (5), 797-800, 2008 | 73 | 2008 |
| Harnessing sulfinyl nitrenes: a unified one-pot synthesis of sulfoximines and sulfonimidamides TQ Davies, MJ Tilby, J Ren, NA Parker, D Skolc, A Hall, F Duarte, ... Journal of the American Chemical Society 142 (36), 15445-15453, 2020 | 68 | 2020 |
| Novel Strategies To Activate the Dopamine D1 Receptor: Recent Advances in Orthosteric Agonism and Positive Allosteric Modulation A Hall, L Provins, A Valade Journal of medicinal chemistry 62 (1), 128-140, 2018 | 64 | 2018 |
| Piperidine-derived γ-secretase modulators A Hall, RL Elliott, GMP Giblin, I Hussain, J Musgrave, A Naylor, R Sasse, ... Bioorganic & Medicinal Chemistry Letters 20 (3), 1306-1311, 2010 | 54 | 2010 |
| Synthesis of hydroxylated pyrrolizidines related to alexine using cycloaddition reactions of functionalised cyclic nitrones A Hall, KP Meldrum, PR Therond, RH Wightman Synlett 1997 (1), 123-125, 1997 | 53 | 1997 |
| γ-Secretase modulators: current status and future directions A Hall, TR Patel Progress in medicinal chemistry 53, 101-145, 2014 | 52 | 2014 |
| The discovery of 6-[2-(5-chloro-2-{[(2, 4-difluorophenyl) methyl] oxy} phenyl)-1-cyclopenten-1-yl]-2-pyridinecarboxylic acid, GW848687X, a potent and selective prostaglandin … GMP Giblin, RA Bit, SH Brown, HM Chaignot, A Chowdhury, IP Chessell, ... Bioorganic & medicinal chemistry letters 17 (2), 385-389, 2007 | 49 | 2007 |
| Discovery of novel, non-acidic 1, 5-biaryl pyrrole EP1 receptor antagonists A Hall, S Atkinson, SH Brown, IP Chessell, A Chowdhury, GMP Giblin, ... Bioorganic & medicinal chemistry letters 17 (5), 1200-1205, 2007 | 46 | 2007 |
| The role of disulfide bond replacements in analogues of the tarantula toxin ProTx-II and their effects on inhibition of the voltage-gated sodium ion channel Nav1. 7 ZVF Wright, S McCarthy, R Dickman, FE Reyes, S Sanchez-Martinez, ... Journal of the American Chemical Society 139 (37), 13063-13075, 2017 | 45 | 2017 |
| -Chloronitroso compounds derived from carbohydrate ketones: cycloadditions with cyclic dienes, a synthesis of ()-physoperuvine and a formal synthesis of (+)-epibatidine A Hall | 45 | 2000 |
| Primary Sulfonamide Synthesis Using the Sulfinylamine Reagent N-Sulfinyl-O-(tert-butyl)hydroxylamine, t-BuONSO TQ Davies, MJ Tilby, D Skolc, A Hall, MC Willis Organic Letters 22 (24), 9495-9499, 2020 | 42 | 2020 |
| Dynamics of Aβ42 reduction in plasma, CSF and brain of rats treated with the γ-secretase modulator, GSM-10h J Hawkins, DC Harrison, S Ahmed, RP Davis, T Chapman, I Marshall, ... Neurodegenerative Diseases 8 (6), 455-464, 2011 | 39 | 2011 |
| Discovery of a novel indole series of EP1 receptor antagonists by scaffold hopping A Hall, A Billinton, SH Brown, A Chowdhury, GMP Giblin, P Goldsmith, ... Bioorganic & medicinal chemistry letters 18 (8), 2684-2690, 2008 | 36 | 2008 |
| Discovery of GSK345931A: An EP1 receptor antagonist with efficacy in preclinical models of inflammatory pain A Hall, SH Brown, C Budd, NM Clayton, GMP Giblin, P Goldsmith, ... Bioorganic & medicinal chemistry letters 19 (2), 497-501, 2009 | 33 | 2009 |
| Identification of novel pyrazole acid antagonists for the EP1 receptor SC McKeown, A Hall, GMP Giblin, O Lorthioir, R Blunt, XQ Lewell, ... Bioorganic & medicinal chemistry letters 16 (18), 4767-4771, 2006 | 33 | 2006 |
| γ‐Secretase modulators do not induce Aβ‐rebound and accumulation of β‐C‐terminal fragment T Li, Y Huang, S Jin, L Ye, N Rong, X Yang, Y Ding, Z Cheng, J Zhang, ... Journal of neurochemistry 121 (2), 277-286, 2012 | 32 | 2012 |
