Segui
Darin E. Jones
Darin E. Jones
Professor of Pharmaceutical Sciences, University of Arkansas for Medical Sciences
Email verificata su uams.edu
Titolo
Citata da
Citata da
Anno
Fourier transform infrared (FTIR) spectroscopy
JS Gaffney, NA Marley, DE Jones
Characterization of Materials, 1-33, 2002
1012002
Design, parallel synthesis, and crystal structures of pyrazinone antithrombotics as selective inhibitors of the tissue factor VIIa complex
JJ Parlow, BL Case, TA Dice, RL Fenton, MJ Hayes, DE Jones, ...
Journal of medicinal chemistry 46 (19), 4050-4062, 2003
972003
Selective small molecule PARG inhibitor causes replication fork stalling and cancer cell death
JH Houl, Z Ye, CA Brosey, LPF Balapiti-Modarage, S Namjoshi, A Bacolla, ...
Nature communications 10 (1), 5654, 2019
912019
Indazole derivatives
IP Buchler, MJ Hayes, SG Hegde, SL Hockerman, DE Jones, SW Kortum, ...
WO Patent 106980, 2009
642009
Structure-based drug design of pyrazinone antithrombotics as selective inhibitors of the tissue factor VIIa complex
MS South, BL Case, RS Wood, DE Jones, MJ Hayes, TJ Girard, ...
Bioorganic & medicinal chemistry letters 13 (14), 2319-2325, 2003
622003
Discovery and SAR of PF-4693627, a potent, selective and orally bioavailable mPGES-1 inhibitor for the potential treatment of inflammation
GB Arhancet, DP Walker, S Metz, YM Fobian, SE Heasley, JS Carter, ...
Bioorganic & medicinal chemistry letters 23 (4), 1114-1119, 2013
562013
Vinyl Oxocarbenium Ions in Intermolecular [4+ 3] Cycloaddition Reactions
M Harmata, DE Jones
The Journal of Organic Chemistry 62 (14), 4885-4885, 1997
551997
Inhibitors of HGFA, matriptase, and hepsin serine proteases: a nonkinase strategy to block cell signaling in cancer
Z Han, PKW Harris, DE Jones, R Chugani, T Kim, M Agarwal, W Shen, ...
ACS medicinal chemistry letters 5 (11), 1219-1224, 2014
522014
Intramolecular [4+ 3] cycloadditions. Studies of relative asymmetric induction
M Harmata, CB Gamlath, CL Barnes, DE Jones
The Journal of Organic Chemistry 60 (16), 5077-5092, 1995
481995
Substituted polycyclic aryl and heteroaryl pyridines useful for selective inhibition of the coagulation cascade
MJ South, B Case, DJ Garland, MJ Hayes, HC Huang, W Huang, ...
US Patent 6,624,180, 2003
462003
Targeting SARS-CoV-2 Nsp3 macrodomain structure with insights from human poly (ADP-ribose) glycohydrolase (PARG) structures with inhibitors
CA Brosey, JH Houl, P Katsonis, LPF Balapiti-Modarage, S Bommagani, ...
Progress in biophysics and molecular biology 163, 171-186, 2021
452021
Intramolecular 4+ 3 cycloadditions. Vinylthionium ions from allylic alcohols
M Harmata, DE Jones
Tetrahedron letters 37 (6), 783-786, 1996
431996
The metallation of Troeger's base
M Harmata, KW Carter, DE Jones, M Kahraman
Tetrahedron letters 37 (35), 6267-6270, 1996
421996
Chiral cations in 4+ 3 cycloadditions
M Harmata, DE Jones, M Kahraman, U Sharma, CL Barnes
Tetrahedron letters 40 (10), 1831-1834, 1999
401999
Structure-based discovery of small molecule hepsin and HGFA protease inhibitors: Evaluation of potency and selectivity derived from distinct binding pockets
FM Franco, DE Jones, PKW Harris, Z Han, SA Wildman, CM Jarvis, ...
Bioorganic & Medicinal Chemistry 23 (10), 2328-2343, 2015
382015
The reaction of N-phenylsulfonimidoyl chloride with trimethylsilylethene. A new route to 2-alkenylanilines
M Harmata, M Kahraman, DE Jones, N Pavri, SE Weatherwax
Tetrahedron 54 (34), 9995-10006, 1998
301998
Nickel Complex Catalyzed Efficient Activation of sp3 and sp2 C–H Bonds for Alkylation and Arylation of Oxygen Containing Heterocyclic Molecules
Y Gartia, P Ramidi, DE Jones, S Pulla, A Ghosh
Catalysis letters 144, 507-515, 2014
292014
Dehydroleucodine, a Sesquiterpene Lactone from Gynoxys verrucosa, Demonstrates Cytotoxic Activity against Human Leukemia Cells
PE Ordóñez, KK Sharma, LM Bystrom, MA Alas, RG Enriquez, O Malagón, ...
Journal of natural products 79 (4), 691-696, 2016
272016
Indazole derivatives as CB1 receptor modulators and their preparation and use in the treatment of CB1-mediated diseases
IP Buchler, MJ Hayes, SG Hedge, SL Hockerman, DE Jones, SW Kortum, ...
Patent WO 106982, 2009
272009
GRB2 enforces homology-directed repair initiation by MRE11
Z Ye, S Xu, Y Shi, A Bacolla, A Syed, D Moiani, CL Tsai, Q Shen, G Peng, ...
Science Advances 7 (32), eabe9254, 2021
262021
Il sistema al momento non può eseguire l'operazione. Riprova più tardi.
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