| A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose JS Tash, B Attardi, SA Hild, R Chakrasali, SR Jakkaraj, GI Georg Biology of reproduction 78 (6), 1127-1138, 2008 | 118 | 2008 |
| Gamendazole, an orally active indazole carboxylic acid male contraceptive agent, targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and stimulates Il1a transcription in rat … JS Tash, R Chakrasali, SR Jakkaraj, J Hughes, SK Smith, K Hornbaker, ... Biology of reproduction 78 (6), 1139-1152, 2008 | 115 | 2008 |
| Development of highly potent and selective diaminothiazole inhibitors of cyclin-dependent kinases E Schonbrunn, S Betzi, R Alam, MP Martin, A Becker, H Han, R Francis, ... Journal of medicinal chemistry 56 (10), 3768-3782, 2013 | 87 | 2013 |
| A Synthesis of 1H-Indazoles via a Cu(OAc)2-Catalyzed N–N Bond Formation C Chen, G Tang, F He, Z Wang, H Jing, R Faessler Organic letters 18 (7), 1690-1693, 2016 | 72 | 2016 |
| Regio-and chemoselective conjugate 1, 4-reduction of α-oxoketene dithioacetals with sodium borohydride and sodium cyanoborohydride CS Rao, RT Chakrasali, H Ila, H Junjappa Tetrahedron 46 (6), 2195-2204, 1990 | 46 | 1990 |
| Regio-and chemoselective conjugate 1, 4-reduction of α-oxoketene dithioacetals with sodium borohydride and sodium cyanoborohydride CS Rao, RT Chakrasali, H Ila, H Junjappa Tetrahedron 46 (6), 2195-2204, 1990 | 46 | 1990 |
| Allosteric indole amide inhibitors of p97: identification of a novel probe of the ubiquitin pathway C Alverez, SL Bulfer, R Chakrasali, MS Chimenti, RJ Deshaies, N Green, ... ACS medicinal chemistry letters 7 (2), 182-187, 2016 | 32 | 2016 |
| Cycloaddition of sodium azide to polarized ketene S, S-and S, N-acetals: synthesis of novel substituted triazole and tetrazole derivatives RT Chakrasali, H Ila, H Junjappa Synthesis 1988 (06), 453-455, 1988 | 26 | 1988 |
| Lonidamine analogues and their use in male contraception and cancer treatment R Chakrasali US Patent US7,514,463, 2009 | 23* | 2009 |
| Lonidamine analogues and their use in male contraception and cancer treatment GI Georg, JS Tash, R Chakrasali, SR Jakkaraj US Patent 7,514,463, 2009 | 23 | 2009 |
| Lonidamine analogues and treatment of polycystic kidney disease IG Georg, JS Tash, R Chakrasali, SR Jakkaraj, JP Calvet US Patent 8,362,031, 2013 | 21 | 2013 |
| Cycloaddition of aroyl/acylketene S, N-acetals with tosyl azide: synthesis of novel 4-aroyl/acyl-5-amino-1H-1, 2, 3-triazoles and 3, 4-annulated 1, 2, 3-triazoles RT Chakrasali, H Ila, H Junjappa Synthesis 1988 (11), 851-854, 1988 | 21 | 1988 |
| Reaction of acylketene S, N-acetals with malonyl chloride: synthesis of novel 1, 5-substituted 4-hydroxy-6-methylthio-2 (1h)-pyridones and 6, 8-substituted 4-hydroxy-7 … RT Chakrasali, H Ila, H Junjappa Synthesis 1988 (1), 87-89, 1988 | 19 | 1988 |
| Total Synthesis and Evaluation of C26-Hydroxyepothilone D Derivatives for Photoaffinity Labeling of β-Tubulin EA Reiff, SK Nair, JT Henri, JF Greiner, BS Reddy, R Chakrasali, ... The Journal of organic chemistry 75 (1), 86-94, 2010 | 16 | 2010 |
| 3-Substituted 1-benzyl-1H-indazole derivatives as antifertility agents B Silvestrini, CY Cheng US Patent 6,001,865, 1999 | 15 | 1999 |
| Reaction of polarized ketene S, N-acetals with bromoacetaldehyde diethyl acetal: synthesis of 1-substituted 3-acyl-and 3-nitro-2-methylthiopyrroles and 1, 2-annulated 3 … AK Gupta, RT Chakrasali, H Ila, H Junjappa Synthesis 2, 141-142, 1989 | 12 | 1989 |
| Discovery of isoxazolyl-based inhibitors of Plasmodium falciparum cGMP-dependent protein kinase SU Mahmood, H Cheng, SR Tummalapalli, R Chakrasali, ... RSC Medicinal Chemistry 11 (1), 98-101, 2020 | 11 | 2020 |
| Cyclocondensation of α‐hydroxyimino‐β‐alkyl/arylimino‐β‐methylthioketones with hydrazine hydrate: Synthesis of 3 (5)‐aryl‐5 (3)‐alkyl/arylamino‐4‐nitroso (or amino) pyrazoles RT Chakrasali, C Srinivasa Rao, H Ila, H Junjappa Journal of heterocyclic chemistry 30 (1), 129-134, 1993 | 10 | 1993 |
| Lonidamine analogues for fertility management IG Georg, JS Tash, R Chakrasali, SR Jakkaraj, K Roby US Patent 8,377,958, 2013 | 7 | 2013 |
| Ila. H.; Junjappa. H A Rahman, RT Chakrasali Indian Journal of Chemistry B 24, 463, 1985 | 6 | 1985 |
Gunda GeorgProfessor of Medicinal Chemistry, University of MinnesotaEmail verificata su umn.edu
