Identification of the spiro (oxindole-3, 3′-thiazolidine)-based derivatives as potential p53 activity modulators I Gomez-Monterrey, A Bertamino, A Porta, A Carotenuto, S Musella, ... Journal of medicinal chemistry 53 (23), 8319-8329, 2010 | 88 | 2010 |
A biomimetic polyketide-inspired approach to small-molecule ligand discovery C Aquino, M Sarkar, MJ Chalmers, K Mendes, T Kodadek, GC Micalizio Nature chemistry 4 (2), 99-104, 2012 | 79 | 2012 |
Synthesis of angularly substituted trans-fused hydroindanes by convergent coupling of acyclic precursors V Jeso, C Aquino, X Cheng, H Mizoguchi, M Nakashige, GC Micalizio Journal of the American Chemical Society 136 (23), 8209-8212, 2014 | 33 | 2014 |
Design, Synthesis, and Cytotoxic Evaluation of Acyl Derivatives of 3-Aminonaphtho[2,3-b]thiophene-4,9-dione, a Quinone-Based System I Gomez-Monterrey, P Campiglia, C Aquino, A Bertamino, I Granata, ... Journal of medicinal chemistry 54 (12), 4077-4091, 2011 | 31 | 2011 |
Design and synthesis of spirotryprostatin-inspired diketopiperazine systems from prolyl spirooxoindolethiazolidine derivatives A Bertamino, C Aquino, M Sala, N de Simone, CA Mattia, L Erra, ... Bioorganic & medicinal chemistry 18 (12), 4328-4337, 2010 | 30 | 2010 |
Spiro[(dihydropyrazin-2,5-dione)-6,3′-(2′,3′-dihydrothieno[2,3-b]naphtho-4′,9′-dione)]-Based Cytotoxic Agents: Structure–Activity Relationship Studies on … I Gomez-Monterrey, P Campiglia, A Carotenuto, P Stiuso, A Bertamino, ... Journal of medicinal chemistry 51 (10), 2924-2932, 2008 | 27 | 2008 |
Spiro[(dihydropyrazin-2,5-dione)-6,3′-(2′,3′-dihydrothieno[2,3-b]naphtho-4′,9′-dione)]-Based Cytotoxic Agents: Structure–Activity Relationship Studies on … I Gomez-Monterrey, P Campiglia, A Carotenuto, P Stiuso, A Bertamino, ... Journal of medicinal chemistry 51 (10), 2924-2932, 2008 | 27 | 2008 |
Recognition of antigen-specific B-cell receptors from chronic lymphocytic leukemia patients by synthetic antigen surrogates M Sarkar, Y Liu, J Morimoto, H Peng, C Aquino, C Rader, N Chiorazzi, ... Chemistry & biology 21 (12), 1670-1679, 2014 | 22 | 2014 |
Decoding split and pool combinatorial libraries with electron-transfer dissociation tandem mass spectrometry M Sarkar, BD Pascal, C Steckler, C Aquino, GC Micalizio, T Kodadek, ... Journal of the American Society for Mass Spectrometry 24 (7), 1026-1036, 2013 | 21 | 2013 |
A novel quinone‐based derivative (DTNQ‐Pro) induces apoptotic death via modulation of heat shock protein expression in Caco‐2 cells I Gomez‐Monterrey, P Campiglia, A Bertamino, C Aquino, M Sala, ... British Journal of Pharmacology 160 (4), 931-940, 2010 | 16 | 2010 |
A New Series of 1,3‐Dihidro‐Imidazo[1,5‐c]thiazole‐5,7‐Dione Derivatives: Synthesis and Interaction with Aβ(25‐35) Amyloid Peptide P Campiglia, M Scrima, M Grimaldi, G Cioffi, A Bertamino, M Sala, ... Chemical biology & drug design 74 (3), 224-233, 2009 | 14 | 2009 |
Synthesis of the cortistatin pentacyclic core by alkoxide-directed metallacycle-mediated annulative cross-coupling C Aquino, SN Greszler, GC Micalizio Organic letters 18 (11), 2624-2627, 2016 | 13 | 2016 |
Novel route in the synthesis of ψ [CH2NH] amide bond surrogate P Campiglia, C Aquino, A Bertamino, M Sala, IM Gomez-Monterrey, ... Tetrahedron Letters 49 (4), 731-734, 2008 | 12 | 2008 |
LiOOt-Bu as a terminal oxidant in a titanium alkoxide-mediated [2+ 2+ 2] reaction cascade WS Kim, C Aquino, H Mizoguchi, GC Micalizio Tetrahedron letters 56 (23), 3557-3559, 2015 | 11 | 2015 |
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based α, α-amino esters P Campiglia, C Aquino, A Bertamino, N De Simone, M Sala, S Castellano, ... Organic & Biomolecular Chemistry 8 (3), 622-627, 2010 | 11 | 2010 |
Synthesis of Novel Indole‐Based Ring Systems by Acid‐Catalysed Condensation from α‐Amino Aldehydes and L‐Trp‐OMe IM Gomez‐Monterrey, P Campiglia, A Bertamino, C Aquino, O Mazzoni, ... European Journal of Organic Chemistry 2008 (11), 1983-1992, 2008 | 5 | 2008 |
(dihydropyrazin-2, 5-Dione)-6, 3′-(2′, 3′-dihydrothieno [2, 3-B] naphtho-4′, 9′-Dione) I Gomez-Monterrey, P Campiglia, A Carotenuto, P Stiuso, A Bertamino, ... Based Cytotoxic Agents: Structure–Activity Relationship Studies on the …, 0 | 4 | |
One Bead-One Compound (OBOC) Peptidomimetic-Encoded Library Synthesis via Split-and-Pool Methods C Aquino, M Sarkar DNA-Encoded Chemical Libraries: Methods and Protocols, 105-120, 2022 | 1 | 2022 |
Kinase modulators and methods of use thereof Z Pei, G Kumar, A Truong, C Aquino, DK Wu, A Tasker US Patent App. 18/210,766, 2024 | | 2024 |
Substituted benzenecarboxamides as il-17a modulators PR Fatheree, MS Linsell, JR Jacobsen, WA VAN DER LINDEN, ... US Patent App. 18/090,319, 2023 | | 2023 |