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Luca Gasparoli
Luca Gasparoli
UCL Institute of Child Health
Verified email at ucl.ac.uk
Title
Cited by
Cited by
Year
hERG1 channels modulate integrin signaling to trigger angiogenesis and tumor progression in colorectal cancer
O Crociani, F Zanieri, S Pillozzi, E Lastraioli, M Stefanini, A Fiore, ...
Scientific reports 3 (1), 3308, 2013
1052013
Potassium channels: novel emerging biomarkers and targets for therapy in cancer
M D'Amico, L Gasparoli, A Arcangeli
Recent patents on anti-cancer drug discovery 8 (1), 53-65, 2013
792013
The combined activation of KCa3. 1 and inhibition of Kv11. 1/hERG1 currents contribute to overcome Cisplatin resistance in colorectal cancer cells
S Pillozzi, M D'Amico, G Bartoli, L Gasparoli, G Petroni, O Crociani, ...
British journal of cancer 118 (2), 200-212, 2018
722018
The conformational state of hERG1 channels determines integrin association, downstream signaling, and cancer progression
A Becchetti, S Crescioli, F Zanieri, G Petroni, R Mercatelli, S Coppola, ...
Science signaling 10 (473), eaaf3236, 2017
612017
NAMI-A is highly cytotoxic toward leukaemia cell lines: Evidence of inhibition of KCa 3.1 channels
S Pillozzi, L Gasparoli, M Stefanini, M Ristori, M D'Amico, E Alessio, ...
Dalton Transactions 43 (32), 12150-12155, 2014
532014
Stromal cell protein kinase C-β inhibition enhances chemosensitivity in B cell malignancies and overcomes drug resistance
E Park, J Chen, A Moore, M Mangolini, A Santoro, JR Boyd, H Schjerven, ...
Science translational medicine 12 (526), eaax9340, 2020
302020
New pyrimido-indole compound CD-160130 preferentially inhibits the KV11. 1B isoform and produces antileukemic effects without cardiotoxicity
L Gasparoli, M D’Amico, M Masselli, S Pillozzi, R Caves, R Khuwaileh, ...
Molecular Pharmacology 87 (2), 183-196, 2015
302015
The AAA+ ATPase RUVBL2 is essential for the oncogenic function of c-MYB in acute myeloid leukemia
E Armenteros-Monterroso, L Zhao, L Gasparoli, T Brooks, K Pearce, ...
Leukemia 33 (12), 2817-2829, 2019
212019
Macrolide antibiotics exert antileukemic effects by modulating the autophagic flux through inhibition of hERG1 potassium channels
S Pillozzi, M Masselli, L Gasparoli, M D'amico, L Polletta, M Veltroni, ...
Blood Cancer Journal 6 (5), e423, 2016
162016
Identification of a c-MYB-directed therapeutic for acute myeloid leukemia
K Clesham, V Walf-Vorderwülbecke, L Gasparoli, C Virely, S Cantilena, ...
Leukemia 36 (6), 1541-1549, 2022
132022
Direct targeted therapy for MLL‐fusion‐driven high‐risk acute leukaemias
S Cantilena, L Gasparoli, D Pal, O Heidenreich, JH Klusmann, ...
Clinical and Translational Medicine 12 (6), e933, 2022
82022
An analytical method for the quantification of hERG1 channel gene expression in human colorectal cancer
A Fortunato, L Gasparoli, S Falsini, B Luca, A Arcangeli
Diagnostic Molecular Pathology 22 (4), 215-221, 2013
52013
ARHGEF4 Regulates an Essential Oncogenic Program in t (12; 21)-Associated Acute Lymphoblastic Leukemia
C Virely, L Gasparoli, M Mangolini, K Clesham, S Inglott, D Edwards, ...
HemaSphere 4 (5), e467, 2020
12020
Targeting ARHGEF4 in cancer
M Mangolini, L Gasparoli, C Virely, D Edwards, J Bartram, N Goulden, ...
Klinische Pädiatrie 229 (03), A5, 2017
12017
Aberrant transcriptional pathways in t(12;21) Acute Lymphoblastic Leukemia
A Sundaresh, L Gasparoli, M Mangolini, D Edwards, M Hubank, T Brooks, ...
Klinische Padiatrie 228 (A12), 2016
12016
Susceptibility of pediatric acute lymphoblastic leukemia to STAT3 inhibition depends on p53 induction
L Gasparoli, C Virely, A Tsakaneli, N Che, D Edwards, J Bartram, ...
Haematologica 109 (4), 1069, 2024
2024
Establishing the mechanism for RUVBL2 essentiality in acute myeloid leukaemia
C Virely, E Armenteros-Monterroso, L Gasparoli, JHA Martens, ...
Klinische Pädiatrie 234 (03), 0011, 2022
2022
Deciphering STAT3 dependency in paediatric acute lymphoblastic leukemia
L Gasparoli, C Virely, S Cantilena, J Bartram, S Inglott, J De Boer, ...
Klinische Pädiatrie 232 (03), 2020
2020
Targeting c-MYB in Acute Leukaemia through Drug Repositioning
KJ Clesham, L Gasparoli, C Virely, S Cantilena, J De Boer, O Williams
Klinische Pädiatrie 231 (03), 38, 2019
2019
hERG1 channel as a molecular target for new anticancer therapeutic approaches
L Gasparoli
2014
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