Synthesis of tryptamine derivatives via a direct, one-pot reductive alkylation of indoles M Righi, F Topi, S Bartolucci, A Bedini, G Piersanti, G Spadoni The Journal of Organic Chemistry 77 (14), 6351-6357, 2012 | 76 | 2012 |
Iridium-catalyzed direct synthesis of tryptamine derivatives from indoles: exploiting N-protected β-amino alcohols as alkylating agents S Bartolucci, M Mari, A Bedini, G Piersanti, G Spadoni The Journal of Organic Chemistry 80 (6), 3217-3222, 2015 | 67 | 2015 |
Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation S Bartolucci, F Bartoccini, M Righi, G Piersanti Organic letters 14 (2), 600-603, 2012 | 41 | 2012 |
Observations concerning the synthesis of tryptamine homologues and branched tryptamine derivatives via the borrowing hydrogen process: synthesis of psilocin, bufotenin, and … S Bartolucci, M Mari, G Di Gregorio, G Piersanti Tetrahedron 72 (18), 2233-2238, 2016 | 39 | 2016 |
Synthesis of Boron‐and Silicon‐Containing Amino Acids through Copper‐Catalysed Conjugate Additions to Dehydroalanine Derivatives F Bartoccini, S Bartolucci, S Lucarini, G Piersanti European Journal of Organic Chemistry 2015 (15), 3352-3360, 2015 | 36 | 2015 |
A simple, modular synthesis of C4-substituted tryptophan derivatives F Bartoccini, S Bartolucci, M Mari, G Piersanti Organic & Biomolecular Chemistry 14 (42), 10095-10100, 2016 | 34 | 2016 |
C4 Pictet–Spengler Reactions for the Synthesis of Core Structures in Hyrtiazepine Alkaloids T Abe, T Haruyama, K Yamada Synthesis 49 (18), 4141-4150, 2017 | 25 | 2017 |
Design, synthesis, and biological activity of hydrogen peroxide responsive arylboronate melatonin hybrids A Bedini, A Fraternale, R Crinelli, M Mari, S Bartolucci, L Chiarantini, ... Chemical Research in Toxicology 32 (1), 100-112, 2018 | 20 | 2018 |
An improved, practical, and scalable five-step synthesis of psilocybin AM Sherwood, P Meisenheimer, G Tarpley, RB Kargbo Synthesis 52 (05), 688-694, 2020 | 19 | 2020 |
Organocatalytic Aza-Friedel–Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho-and Benzofuranones Bearing a Quaternary Center at … F Bartoccini, M Mari, M Retini, S Bartolucci, G Piersanti The Journal of Organic Chemistry 83 (19), 12275-12283, 2018 | 19 | 2018 |
Concise and convergent enantioselective total syntheses of (+)-and (−)-fumimycin M Retini, S Bartolucci, F Bartoccini, M Mari, G Piersanti The Journal of Organic Chemistry 84 (18), 12221-12227, 2019 | 18 | 2019 |
Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation G Di Gregorio, M Mari, S Bartolucci, F Bartoccini, G Piersanti Organic Chemistry Frontiers 5 (10), 1622-1627, 2018 | 15 | 2018 |
Synthesis and configuration determination of all enantiopure stereoisomers of the melatonin receptor ligand 4-phenyl-2-propionamidotetralin using an expedient optical … S Lucarini, S Bartolucci, A Bedini, G Gatti, P Orlando, G Piersanti, ... Organic & Biomolecular Chemistry 10 (2), 305-313, 2012 | 13 | 2012 |
Chiral recognition of flexible melatonin receptor ligands induced by conformational equilibria GM Elisi, A Bedini, L Scalvini, C Carmi, S Bartolucci, V Lucini, F Scaglione, ... Molecules 25 (18), 4057, 2020 | 10 | 2020 |
Synthesis and Characterization of New Bivalent Agents as Melatonin- and Histamine H3-Ligands D Pala, L Scalvini, A Lodola, M Mor, L Flammini, E Barocelli, V Lucini, ... International Journal of Molecular Sciences 15 (9), 16114-16133, 2014 | 10 | 2014 |
Reductive N-arylethylation of aromatic amines and N-heterocycles with enol ethers K Vögerl, DN Ong, F Bracher Synthesis 50 (06), 1323-1330, 2018 | 9 | 2018 |
Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties G Spadoni, A Bedini, S Bartolucci, D Pala, M Mor, T Riccioni, F Borsini, ... European Journal of Medicinal Chemistry 80, 8-35, 2014 | 8 | 2014 |
N‐(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability F Ferlenghi, M Mari, G Gobbi, GM Elisi, M Mor, S Rivara, F Vacondio, ... ChemMedChem 16 (19), 3071-3082, 2021 | 6 | 2021 |
Recent advances in the applications of triethylsilane in organic synthesis V Ručilová, M Soural Synthesis 50 (19), 3809-3824, 2018 | 6 | 2018 |
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H‐Bond‐Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α‐Amino Acids M Retini, S Bartolucci, F Bartoccini, G Piersanti Chemistry–A European Journal 28 (57), e202201994, 2022 | 2 | 2022 |