Tanja Schirmeister
Tanja Schirmeister
University of Mainz, Pharmacy, Prof. Pharm. Med. Chem.
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Cysteine proteases and their inhibitors
HH Otto, T Schirmeister
Chemical reviews 97 (1), 133-172, 1997
Development of peptidomimetics with a vinyl sulfone warhead as irreversible falcipain-2 inhibitors
R Ettari, E Nizi, ME Di Francesco, MA Dude, G Pradel, R Vičík, ...
Journal of medicinal chemistry 51 (4), 988-996, 2008
Biochemistry and medicinal chemistry of the dengue virus protease
C Nitsche, S Holloway, T Schirmeister, CD Klein
Chemical reviews 114 (22), 11348-11381, 2014
Novel dengue virus NS2B/NS3 protease inhibitors
H Wu, S Bock, M Snitko, T Berger, T Weidner, S Holloway, M Kanitz, ...
Antimicrobial agents and chemotherapy 59 (2), 1100-1109, 2015
Flavonoids as noncompetitive inhibitors of Dengue virus NS2B-NS3 protease: Inhibition kinetics and docking studies
LRF de Sousa, H Wu, L Nebo, JB Fernandes, W Kiefer, M Kanitz, ...
Bioorganic & medicinal chemistry 23 (3), 466-470, 2015
Prospective evaluation of free energy calculations for the prioritization of Cathepsin L inhibitors
B Kuhn, M Tichý, L Wang, S Robinson, RE Martin, A Kuglstatter, J Benz, ...
Journal of medicinal chemistry 60 (6), 2485-2497, 2017
Transcriptome and functional analysis of the eukaryotic-type serine/threonine kinase PknB in Staphylococcus aureus
S Donat, K Streker, T Schirmeister, S Rakette, T Stehle, M Liebeke, M Lalk, ...
Journal of bacteriology 191 (13), 4056-4069, 2009
Inhibitors of cysteine proteases
R Vicik, M Busemann, K Baumann, T Schirmeister
Current topics in medicinal chemistry 6 (4), 331-353, 2006
The significance of ionic bonding in sulfur dioxide: Bond orders from X‐ray diffraction data
S Grabowsky, P Luger, J Buschmann, T Schneider, T Schirmeister, ...
Angewandte Chemie International Edition 27 (51), 6776-6779, 2012
Aziridine-2,3-dicarboxylate inhibitors targeting the major cysteine protease of Trypanosoma brucei as lead trypanocidal agents
R Vicik, V Hoerr, M Glaser, M Schultheis, E Hansell, JH McKerrow, ...
Bioorganic & medicinal chemistry letters 16 (10), 2753-2757, 2006
Antioxidant and anti-protease activities of diazepinomicin from the sponge-associated Micromonospora strain RV115
UR Abdelmohsen, M Szesny, EM Othman, T Schirmeister, S Grond, ...
Marine drugs 10 (10), 2208-2221, 2012
Allicin and derivates are cysteine protease inhibitors with antiparasitic activity
T Waag, C Gelhaus, J Rath, A Stich, M Leippe, T Schirmeister
Bioorganic & medicinal chemistry letters 20 (18), 5541-5543, 2010
Aziridine-2, 3-dicarboxylates, peptidomimetic cysteine protease inhibitors with antileishmanial activity
A Ponte-Sucre, R Vicik, M Schultheis, T Schirmeister, H Moll
Antimicrobial agents and chemotherapy 50 (7), 2439-2447, 2006
Novel peptidomimetics containing a vinyl ester moiety as highly potent and selective falcipain-2 inhibitors
R Ettari, N Micale, T Schirmeister, C Gelhaus, M Leippe, E Nizi, ...
Journal of medicinal chemistry 52 (7), 2157-2160, 2009
New peptidic cysteine protease inhibitors derived from the electrophilic α-amino acid aziridine-2, 3-dicarboxylic acid
T Schirmeister
Journal of medicinal chemistry 42 (4), 560-572, 1999
Metabolomics analysis and biological investigation of three Malvaceae plants
OH Abdelhafez, EM Othman, JR Fahim, SY Desoukey, ...
Phytochemical Analysis 31 (2), 204-214, 2020
Evidence for substrate binding-induced zwitterion formation in the catalytic Cys-His dyad of the SARS-CoV main protease
A Paasche, A Zipper, S Schäfer, J Ziebuhr, T Schirmeister, B Engels
Biochemistry 53 (37), 5930-5946, 2014
Aziridinyl peptides as inhibitors of cysteine proteases: effect of a free carboxylic acid function on inhibition
T Schirmeister, M Peric
Bioorganic & medicinal chemistry 8 (6), 1281-1291, 2000
A new lead for nonpeptidic active-site-directed inhibitors of the severe acute respiratory syndrome coronavirus main protease discovered by a combination of screening and …
U Kaeppler, N Stiefl, M Schiller, R Vicik, A Breuning, W Schmitz, ...
Journal of medicinal chemistry 48 (22), 6832-6842, 2005
Quantum chemical-based protocol for the rational design of covalent inhibitors
T Schirmeister, J Kesselring, S Jung, TH Schneider, A Weickert, J Becker, ...
Journal of the American Chemical Society 138 (27), 8332-8335, 2016
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