Fabrizio Manetti
Fabrizio Manetti
Associate Professor, University of Siena (Italy)
Verified email at unisi.it
Title
Cited by
Cited by
Year
MmpL3 is the cellular target of the antitubercular pyrrole derivative BM212
V La Rosa, G Poce, JO Canseco, S Buroni, MR Pasca, M Biava, RM Raju, ...
Antimicrobial agents and chemotherapy 56 (1), 324-331, 2012
1822012
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones
D Castagnolo, F Manetti, M Radi, B Bechi, M Pagano, A De Logu, ...
Bioorganic & medicinal chemistry 17 (15), 5716-5721, 2009
1662009
Synthesis, Biological Evaluation, and Pharmacophore Generation of New Pyridazinone Derivatives with Affinity toward α1-and α2-Adrenoceptors 1
R Barbaro, L Betti, M Botta, F Corelli, G Giannaccini, L Maccari, F Manetti, ...
Journal of medicinal chemistry 44 (13), 2118-2132, 2001
1382001
Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis
D Castagnolo, A De Logu, M Radi, B Bechi, F Manetti, M Magnani, ...
Bioorganic & medicinal chemistry 16 (18), 8587-8591, 2008
1332008
Antimycobacterial agents. Novel diarylpyrrole derivatives of BM212 endowed with high activity toward Mycobacterium tuberculosis and low cytotoxicity
M Biava, GC Porretta, G Poce, S Supino, D Deidda, R Pompei, P Molicotti, ...
Journal of medicinal chemistry 49 (16), 4946-4952, 2006
1182006
Fibroblast growth factors and their inhibitors
F Manetti, F Corelli, M Botta
Current pharmaceutical design 6 (18), 1897-1924, 2000
1052000
LIM kinases are attractive targets with many macromolecular partners and only a few small molecule regulators
F Manetti
Medicinal research reviews 32 (5), 968-998, 2012
1002012
Antifungal Agents. 10. New Derivatives of 1-[(Aryl)[4-aryl-1 H-pyrrol-3-yl] methyl]-1 H-imidazole, Synthesis, Anti-Candida Activity, and Quantitative Structure-Analysis …
A Tafi, R Costi, M Botta, R Di Santo, F Corelli, S Massa, A Ciacci, ...
Journal of medicinal chemistry 45 (13), 2720-2732, 2002
992002
New pyrazolo [3, 4-d] pyrimidines endowed with A431 antiproliferative activity and inhibitory properties of Src phosphorylation
S Schenone, O Bruno, A Ranise, F Bondavalli, C Brullo, P Fossa, L Mosti, ...
Bioorganic & medicinal chemistry letters 14 (10), 2511-2517, 2004
972004
Antimycobacterial compounds. New pyrrole derivatives of BM212
M Biava, GC Porretta, D Deidda, R Pompei, A Tafi, F Manetti
Bioorganic & medicinal chemistry 12 (6), 1453-1458, 2004
962004
Pyrazolo [3, 4-d] pyrimidines as potent antiproliferative and proapoptotic agents toward A431 and 8701-BC cells in culture via inhibition of c-Src phosphorylation
F Carraro, A Naldini, A Pucci, GA Locatelli, G Maga, S Schenone, O Bruno, ...
Journal of medicinal chemistry 49 (5), 1549-1561, 2006
942006
Computational comparison of microtubule-stabilising agents laulimalide and peloruside with taxol and colchicine
O Pineda, J Farrąs, L Maccari, F Manetti, M Botta, J Vilarrasa
Bioorganic & medicinal chemistry letters 14 (19), 4825-4829, 2004
902004
Importance of the thiomorpholine introduction in new pyrrole derivatives as antimycobacterial agents analogues of BM 212
M Biava, GC Porretta, D Deidda, R Pompei, A Tafi, F Manetti
Bioorganic & medicinal chemistry 11 (4), 515-520, 2003
882003
Structure-based optimization of pyrazolo [3, 4-d] pyrimidines as Abl inhibitors and antiproliferative agents toward human leukemia cell lines
F Manetti, C Brullo, M Magnani, F Mosci, B Chelli, E Crespan, ...
Journal of medicinal chemistry 51 (5), 1252-1259, 2008
842008
Pharmacophore Modeling and Molecular Docking Led to the Discovery of Inhibitors of Human Immunodeficiency Virus-1 Replication Targeting the Human Cellular Aspartic Acid …
G Maga, F Falchi, A Garbelli, A Belfiore, M Witvrouw, F Manetti, M Botta
Journal of medicinal chemistry 51 (21), 6635-6638, 2008
822008
1, 5-Diphenylpyrrole derivatives as antimycobacterial agents. Probing the influence on antimycobacterial activity of lipophilic substituents at the phenyl rings
M Biava, GC Porretta, G Poce, A De Logu, M Saddi, R Meleddu, F Manetti, ...
Journal of medicinal chemistry 51 (12), 3644-3648, 2008
822008
Identification of a Novel Pyrazolo[3,4-d]pyrimidine Able To Inhibit Cell Proliferation of a Human Osteogenic Sarcoma in Vitro and in a Xenograft Model in Mice
F Manetti, A Santucci, GA Locatelli, G Maga, A Spreafico, T Serchi, ...
Journal of medicinal chemistry 50 (23), 5579-5588, 2007
822007
Synthesis, biological evaluation and docking studies of 4-amino substituted 1H-pyrazolo [3, 4-d] pyrimidines
S Schenone, C Brullo, O Bruno, F Bondavalli, L Mosti, G Maga, E Crespan, ...
European journal of medicinal chemistry 43 (12), 2665-2676, 2008
812008
Antiproliferative activity of new 1-aryl-4-amino-1H-pyrazolo [3, 4-d] pyrimidine derivatives toward the human epidermoid carcinoma A431 cell line
S Schenone, O Bruno, F Bondavalli, A Ranise, L Mosti, G Menozzi, ...
European journal of medicinal chemistry 39 (11), 939-946, 2004
802004
Acylthiourea, acylurea, and acylguanidine derivatives with potent hedgehog inhibiting activity
A Solinas, H Faure, H Roudaut, E Traiffort, A Schoenfelder, A Mann, ...
Journal of medicinal chemistry 55 (4), 1559-1571, 2012
792012
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