| Discovery of a potential allosteric ligand binding site in CDK2 S Betzi, R Alam, M Martin, DJ Lubbers, H Han, SR Jakkaraj, GI Georg, ... ACS chemical biology 6 (5), 492-501, 2011 | 188 | 2011 |
| A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose JS Tash, B Attardi, SA Hild, R Chakrasali, SR Jakkaraj, GI Georg Biology of reproduction 78 (6), 1127-1138, 2008 | 118 | 2008 |
| Gamendazole, an orally active indazole carboxylic acid male contraceptive agent, targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and stimulates Il1a transcription in rat … JS Tash, R Chakrasali, SR Jakkaraj, J Hughes, SK Smith, K Hornbaker, ... Biology of reproduction 78 (6), 1139-1152, 2008 | 115 | 2008 |
| Development of highly potent and selective diaminothiazole inhibitors of cyclin-dependent kinases E Schonbrunn, S Betzi, R Alam, MP Martin, A Becker, H Han, R Francis, ... Journal of medicinal chemistry 56 (10), 3768-3782, 2013 | 87 | 2013 |
| Lonidamine analogues and their use in male contraception and cancer treatment GI Georg, JS Tash, R Chakrasali, SR Jakkaraj US Patent 7,514,463, 2009 | 23 | 2009 |
| Lonidamine analogues and treatment of polycystic kidney disease IG Georg, JS Tash, R Chakrasali, SR Jakkaraj, JP Calvet US Patent 8,362,031, 2013 | 21 | 2013 |
| Scalable syntheses of the BET bromodomain inhibitor JQ1 SS Syeda, S Jakkaraj, GI Georg Tetrahedron letters 56 (23), 3454-3457, 2015 | 19 | 2015 |
| Synthesis and antibacterial activity of 6-aryl-3-(2′-methyl-1′, 8′-naphthyridin-3′-yl)-1, 2, 4-triazolo-[3, 4-b][1, 3, 4] thiadiazoles HS Rani, K Mogilaiah, JS Rao, B Sreenivasulu Indian Journal of Chemistry-Section B Organic and Medicinal Chemistry 35 (7 …, 1996 | 11 | 1996 |
| Syntheses of PDE3A inhibitor ORG9935 and determination of the absolute stereochemistries of its enantiomers by X-ray crystallography SR Jakkaraj, VG Young Jr, GI Georg Tetrahedron 74 (22), 2769-2774, 2018 | 8 | 2018 |
| N-Butyldeoxygalactonojirimycin Induces Reversible Infertility in Male CD Rats V Gupta, SA Hild, SR Jakkaraj, EJ Carlson, HL Wong, CL Allen, GI Georg, ... International Journal of Molecular Sciences 21 (1), 301, 2019 | 7 | 2019 |
| Lonidamine analogues for fertility management IG Georg, JS Tash, R Chakrasali, SR Jakkaraj, K Roby US Patent 8,377,958, 2013 | 7 | 2013 |
| Lonidamine analogues for fertility management IG Georg, JS Tash, R Chakrasali, SR Jakkaraj, K Roby US Patent 8,377,958, 2013 | 7 | 2013 |
| Synthesis of 2-(3-aryl-4-formylpyrazol-1-yl)-3-phenyl-1, 8-naphthyridines JS Rao, K Mogilaiah, B Sreenivasulu Indian Journal of Chemistry-Section B Organic and Medicinal Chemistry 35 (7 …, 1996 | 6 | 1996 |
| Anti-Spermatogenic Efficacy of Nonhormonal Male Contraceptive Agent, H2-Gamendazole, in Mice, Rats, Rabbits, and Nonhuman Primates (Rhesus), and a Multiple Low Dose Oral … VG Gupta, M Zelinski, K Steinmetz, A Miklos, M Broward, S Jakkaraj, ... Biology of Reproduction 85 (Suppl_1), 5-5, 2011 | 3 | 2011 |
| Synthesis of pyrazole-1-carbonyl-1,8-naphthyridines as antimicrobial agents KM J. Sudhakar Rao, B. Sreenivasulu Indian Journal of Chemistry 26 (44), 734, 1995 | 3* | 1995 |
| The orally active male contraceptive agent H2‐gamendazole interacts with organic anion transporting polypeptides expressed in human hepatocytes (1064.18) J Shoop, L Holets, S Jakkaraj, G Georg, C Flynn, M Baltezor, J Tash, ... The FASEB Journal 28, 1064.18, 2014 | 2 | 2014 |
| The lonidamine derivative H2-gamendazole reduces cyst formation in polycystic kidney disease SV Sundar, JX Zhou, BS Magenheimer, GA Reif, DP Wallace, GI Georg, ... American Journal of Physiology-Renal Physiology 323 (4), F492-F506, 2022 | 1 | 2022 |
| Effect of H2-Gamendazole and Other Indazole Carboxylic Acid (ICA) Analogs on Primary Rat Sertoli Cells Cytoskeletal Structure and Elongation Factor 1 Alpha (EEF1A1) Expression … LM Holets, J Cottita, S Jakkaraj, R Chakrasali, T Kinzy, G Georg, J Tash Biology of Reproduction 85 (Suppl_1), 582-582, 2011 | 1 | 2011 |
| In Vitro Versus In Vivo Effects of NB-DGJ and NB-DNJ as Lead Compounds for Development of Non-Hormonal Reversible Oral Male Contraceptives. VG Gupta, S Hild, S Jakkaraj, GI Georg, JS Tash Biology of Reproduction 83 (Suppl_1), 679-679, 2010 | 1 | 2010 |
| Synthesis of some 31-(2-methyl-1,8-naphthyridine-3-carbonylamino)spiro-[3H-indole-3,21-thiazolidine)-2,41(1H)-diones and 2-(2-methyl-1,8-naphthyridin-3-yl)-(1,3,4)-oxadiazino … BS 11. H. Shailaja Rani, K. Mogilaiah, J. Sudhakar Rao Indian Journal of Chemistry, 1035, 1995 | 1 | 1995 |
